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Citations for Tocris :
51 - 100 of 1908 citations for 6H Pyrazolo 3 4 b pyridin 6 one 3 cyclobutyl 1 2 4 5 tetrahydro 4 methyl 9CI since 2019
Citations are collected from bioRxiv only, the total number of publications could be much larger.
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bioRxiv - Neuroscience 2020Quote: ... Readings were taken before and 3–4 min after application of 20 μM 2-AG (Tocris) to activate CB1R or the eCB sensor.
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bioRxiv - Neuroscience 2020Quote: ... The GAT1 blocker NO-711 [(1,2,5,6-tetrahydro-1-[2-[[(diphenylmethylene)amino]oxy]ethyl]-3-pyridinecarboxylic acid hydrochloride] and GAT3 blocker SNAP-5114 [1-[2-[tris(4-methoxyphenyl)methoxy]ethyl]-(S)-3-piperidinecarboxylic acid] were purchased from Tocris Bioscience (Minneapolis ...
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bioRxiv - Neuroscience 2022Quote: ... 3,5-dichloro-N-[[(1α,5α,6-exo,6α)-3-(3,3-dimethylbutyl)-3-azabicyclo[3.1.0]hex-6-yl]methyl]-benzamide-hydrochloride (ML218 or ml) was purchased from TOCRIS and initially dissolved at 50 mM in DMSO ...
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bioRxiv - Neuroscience 2023Quote: ... (αR,βS)-α-(4-Hydroxyphenyl)-β-methyl-4-(phenylmethyl)-1-piperidinepropanol maleate (Ro25-6981, 1 μM dissolved in H2O; Tocris Bioscience), 5-(4-Bromophenyl)-3-(1,2-dihydro-6-methyl-2-oxo-4-phenyl-3-quinolinyl)-4,5-dihydro-γ-oxo-1H-pyrazole-1-butanoic acid (DQP 1105 ...
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bioRxiv - Cell Biology 2021Quote: 4-Methoxy-3-(2-phenylethoxy)-N,N-dipropylbenzeneethanamine hydrochloride (NE-100 hydrochloride) was purchased from Tocris (3133). Stock and work solutions were prepared using 100% dimethyl sulfoxide sterile-filtered (DMSO ...
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bioRxiv - Neuroscience 2024Quote: ... 4-(2-Butyl-6,7-dichloro-2-cyclopentyl-indan-1-on-5-yl) oxobutyric acid (DCPIB; Tocris), superoxide dismutase (SOD ...
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bioRxiv - Cell Biology 2021Quote: ... interleukin-1 receptor-associated kinase 1 and 4 (IRAK 1/4; IRAK 1/4 inhibitor, 0.1 μM; Tocris); TANK-binding kinase 1 (TBK1 ...
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bioRxiv - Cancer Biology 2021Quote: ... 4 μM IWP-2 (Tocris), and 1 μM A83-01 (Tocris) ...
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bioRxiv - Neuroscience 2019Quote: ... yohimbine (2–4 µM; Tocris). Endogenous dopamine levels were manipulated with the DAT inhibitor GBR-12909 (10 µM ...
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bioRxiv - Developmental Biology 2020Quote: ... 4 μM IWP-2 (Tocris), and 1 μM A83-01 (Tocris ...
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bioRxiv - Neuroscience 2019Quote: ... and substracted from background noise by detecting events in the last 4 seconds of 5 EPSCs at 0.2 Hz in 3 mM NBQX (Tocris) in extracellular solution.
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Dopamine depletion can be predicted by the aperiodic component of subthalamic local field potentialsbioRxiv - Neuroscience 2021Quote: ... 4 or 8 μl of 6-OHDA (5 μg in 1 μl saline containing 0.1% ascorbic acid; Tocris, Bristol ...
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bioRxiv - Developmental Biology 2022Quote: 4-Hydroxytamoxifen (4-OHT) (Tocris Bioscience) was dissolved in corn oil (Millipore-Sigma ...
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bioRxiv - Neuroscience 2022Quote: ... was inserted into the guide cannula and a Hamilton Syringe was used to administrate 1 μL of 2 mM pyridoxalphosphate-6-azophenyl-2’,4’-disulfonic acid (PPADS, Tocris, 0625), 1.5 μg/μL S961 (Phoenix Pharmaceuticals ...
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bioRxiv - Immunology 2023Quote: ... 49 µM of TLR 4/6 inhibitor (GIT27, Tocris) or 10 µM of TLR 8 inhibitor (Cu-CPT9a ...
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bioRxiv - Neuroscience 2020Quote: ... medium was exchanged every 3-4 days with RGC induction media containing: DAPT (3uM, Tocris), 10μM Rock inhibitor (Y27632) ...
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bioRxiv - Neuroscience 2023Quote: ... 2 CaCl2 and 4 MNI-glutamate (Tocris). aCSF was continually bubbled with 95%O2 and 5%CO2 ...
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bioRxiv - Neuroscience 2019Quote: ... (3S)-3-[[3-[[4-(Trifluoromethyl)benzoyl]amino]phenyl]methoxy]-L-aspartic acid (TFB-TBOA) was purchased from Tocris (Minneapolis, MN; Cat# 2532). All other chemicals were purchased from MilliporeSigma (Burlington ...
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bioRxiv - Neuroscience 2023Quote: The neural activity was reversibly suppressed using the GABA-A agonist 4,5,6,7-tetrahydro isoxazole [5,4-c]-pyridine-3-ol (THIP hydrochloride; Tocris). The THIP was dissolved in phosphate-buffered saline (PBS) ...
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bioRxiv - Neuroscience 2020Quote: MPEP (2-Methyl-6-(phenylethynyl)pyridine) from Tocris
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bioRxiv - Neuroscience 2020Quote: ... 4-aminopyrimidine (4-ap, 30 µM, Tocris) and/or Tetrodotoxin (TTX ...
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bioRxiv - Neuroscience 2020Quote: ... 100 4-aminopyridine (4-AP) (Tocris Bioscience). To determine possible changes in intrinsic excitability ...
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bioRxiv - Biophysics 2022Quote: ... or 4 μM GsMTx-4 (Tocris 4912) were incubated for 15 min ...
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bioRxiv - Neuroscience 2023Quote: ... 100 μM 4-aminopyridin (4-AP, Tocris) and 20 mM tetraethylammonium chloride (TEA ...
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bioRxiv - Neuroscience 2023Quote: ... and (3-chloro-4-fluoro-N-[(4-([2-(phenylcarbonyl)hydrazino]carbonyl) phenyl)methyl]benzene-sulfonamide) (TCN-201) (Hansen et al., 2012)were obtained from Tocris Bioscience ...
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bioRxiv - Neuroscience 2019Quote: ... (9S,10R,12R)-2,3,9,10,11,12-Hexahydro-10-hydroxy-9-methyl-1-oxo-9,12-epoxy-1H-diindolo[1,2,3-fg:3’,2’,1’-kl]pyrrolo[3,4-i][1,6]benzodiazocine-10-carboxylic acid methyl ester (K252a, 200 nM) (Tocris), 7,8-Dihydroxy-2-phenyl-4H-1-benzopyran-4-one (DHF ...
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bioRxiv - Microbiology 2022Quote: NADA (3-[(7-Nitro-2,1,3-benzoxadiazol-4-yl)amino]-D-alanine hydrochloride) was synthesized by Tocris following the published protocol (31) ...
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bioRxiv - Neuroscience 2023Quote: ... 4-AP (10 μM, Tocris, #504-24-5), Phenytoin (25 μM ...
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bioRxiv - Neuroscience 2023Quote: ... in combination with potassium channel blocker 4-aminopyridine (4-AP, 1 mM, Tocris) to facilitate transmitter release at monosynaptic connections from RSC to ChC and recorded the PSP amplitudes (Figure 1H) ...
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bioRxiv - Neuroscience 2019Quote: ... (+)-4-[(αR)-α-((2S,5R)-4-Allyl-2,5-dimethyl-1-piperazinyl)-3-methoxybenzyl]-N,N-diethylbenzamide (SNC 80) (20mg/kg; Tocris) dissolved in 1mM HCl in saline.
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bioRxiv - Neuroscience 2022Quote: 5-[2-Chloro-6-(trifluoromethoxy)phenyl]-1,3-dihydro-2H-benzimidazol-2-one (JNJ-5; Tocris, Minneapolis, MN) is a high affinity ...
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bioRxiv - Neuroscience 2019Quote: ... and 20 mM 4-aminopyridine (4-AP; Tocris) were included for more stringent isolation of monosynaptic transmission (Cruikshank et al. ...
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bioRxiv - Pharmacology and Toxicology 2021Quote: ... N,N’-Dicyclohexylcarbamimidothioic acid (5,6-dihydro-6,6-dimethylimidazo[2,1-b]thiazol-3-yl)methyl ester dihydrochloride (IT1t) was purchased from Tocris (United Kingdom). Bovine serum albumin ...
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bioRxiv - Neuroscience 2020Quote: ... exendin-4 (Tocris, 1 mg/mL), or y-msh (Tocris ...
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bioRxiv - Neuroscience 2020Quote: ... PSB0739 (4 hours, 1 μM, Tocris) or MRS2211 (4 hours ...
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bioRxiv - Neuroscience 2020Quote: ... or 4-aminopyridine (4-AP, Cat. No. 0940, Tocris), diluted in culture medium at a final concentration of 1 μM and 50 μM ...
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bioRxiv - Neuroscience 2023Quote: ... 4-Aminopyridine (4- AP; 100 µM; Tocris, Item# 0940), 6,7-Dinitroquinoxaline-2,3-dione (DNQX ...
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bioRxiv - Cell Biology 2021Quote: ... CBA (4-chloro-2-[[2-(2-chlorophenoxy) acetyl aminobenzoic acid from Tocris Bioscience (Minneapolis ...
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bioRxiv - Microbiology 2023Quote: ... cells were resuspended in 25 µl PBS together with 0.25 µl of 5 mM 3-[[(7-Hydroxy-2-oxo-2H-1-benzopyran-3-yl) carbonyl]amino]-D-alanine hydrocholoride (HADA) (Tocris) dissolved in DMSO ...
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bioRxiv - Neuroscience 2024Quote: ... CACNA1A+/− networks on MEA at DIV51 were treated with 20 µM 4-aminopyridine (4-AP; Tocris, #504-24-5) and recorded for 30 minutes after the compound was added ...
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bioRxiv - Molecular Biology 2022Quote: Parental A549 cells were fixed with 4% paraformaldehyde following 3-hour treatment with poly I:C (2.0 μg/mL, Tocris), LPS (1.0 μg/mL ...
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Pathogenic CD8 T cell responses are driven by neutrophil-mediated hypoxia in cutaneous leishmaniasisbioRxiv - Immunology 2023Quote: ... the sections were counter-stained with the nuclear probe 4’,6-diamino-2-phenylindole (DAPI, Biotechne-Tocris, UK). Slides were covered with Prolong™ Gold Antifade Mountant (Invitrogen ...
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bioRxiv - Cell Biology 2022Quote: ... 1,1-Dimethyl-4-diphenylacetoxypiperidinium iodide (4-DAMP, 0.1 µM, Tocris), U73122 (10 µM ...
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bioRxiv - Neuroscience 2021Quote: ... and 4-AP (1 mM, Tocris Bioscience), as was done previously (Carta et al. ...
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bioRxiv - Developmental Biology 2023Quote: ... 1 µM 4-OH-TMX (Tocris Bioscience) was added to sustain knockout efficiency ...
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bioRxiv - Immunology 2019Quote: ... 4-Hydroxytamoxifen (Tocris), CFSE (BioLegend) ...
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bioRxiv - Neuroscience 2022Quote: ... Exendin-4 (Tocris) was administered at 0.004 to 0.04 mg/kg ...
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bioRxiv - Neuroscience 2022Quote: ... DSP-4 (Tocris) was dissolved in saline and a single dose (75 mg/kg BW ...
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bioRxiv - Neuroscience 2023Quote: ... 4-AP (100 µM, Tocris, 0940, CAS: 504-24-5), CNQX (20 µM ...
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bioRxiv - Biochemistry 2024Quote: ... The filtrate was diluted two times the volume with buffer UA (8 M urea [Acros Organics, CAS No. 57-13-6], 50 mM sodium acetate [Tocris CAS No. 127-09-3], pH 4). This was loaded onto a HiPrep SP HP 16/10 (Cytiva ...