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Citations for Tocris :
51 - 100 of 772 citations for 6 Hydroxy 2 2 pyridinyl 4 3H pyrimidinone since 2019
Citations are collected from bioRxiv only, the total number of publications could be much larger.
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bioRxiv - Pharmacology and Toxicology 2023Quote: ... [2-Amino-4-[3-(trifluoromethyl)phenyl]-3-thienyl] phenylmethanone (VCP 171; Tocris, 1018830-99-3), 5-[2-(5-nitro-2-furanyl)ethenyl]-2-furancarboxylic acid ...
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bioRxiv - Cell Biology 2021Quote: ... 2-APB (Tocris), Xestospongin C (Tocris) ...
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bioRxiv - Neuroscience 2020Quote: ... co-applied with the competitive α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid AMPA/kainate receptor antagonist CNQX (Tocris; 20 μM) (n=13) ...
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bioRxiv - Neuroscience 2023Quote: ... 3-Chloro-4-fluoro-N-[4-[[2-(phenylcarbonyl) hydrazino]carbonyl]benzyl]benzene-sulfonamide (TCN 201, 3 μM dissolved in DMSO; Tocris Bioscience), (αR,βS)-α-(4-Hydroxyphenyl)-β-methyl-4-(phenylmethyl)-1-piperidinepropanol maleate (Ro25-6981 ...
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bioRxiv - Cell Biology 2022Quote: ... The FFA2R antagonist CATPB ((S)-3-(2-(3-chlorophenyl)acetamido)-4-(4-(trifluoromethyl)-phenyl) butanoic acid) was from Tocris (Britsol, UK).
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bioRxiv - Immunology 2022Quote: ... 2-aminoethoxydiphenyl borate (2-APB) or trans-Ned-19 (all Tocris).
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bioRxiv - Animal Behavior and Cognition 2022Quote: ... (R)-(+)-WIN 55,212-2) WIN 55,212-2 was purchased from Tocris Cookson Ltd ...
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bioRxiv - Biochemistry 2023Quote: ... 5% CO2 with either DMSO or MLi-2 (Tocris; 2 μM) for 1 hour ...
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bioRxiv - Immunology 2023Quote: ... 49 µM of TLR 4/6 inhibitor (GIT27, Tocris) or 10 µM of TLR 8 inhibitor (Cu-CPT9a ...
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bioRxiv - Neuroscience 2020Quote: ... Readings were taken before and 3–4 min after application of 20 μM 2-AG (Tocris) to activate CB1R or the eCB sensor.
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bioRxiv - Neuroscience 2021Quote: ... 6R)-4-Amino-2-oxabicyclo [3.1.0] hexane-4,6-dicarboxylic acid disodium salt (LY379268, 100 µM, Tocris); calmidazolium chloride (CMZ ...
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bioRxiv - Neuroscience 2024Quote: ... The following competitive antagonists were employed for microscopical experiments: trans-2-Carboxy-5,7-dichloro-4-phenylaminocarbonylamino-1,2,3,4-tetrahydroquinoline (L-689-560; Tocris); 7-Chloro-4-hydroxy-3-(3-phenoxy)phenyl-2(1H)-quinolinone (L-701-324 ...
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bioRxiv - Neuroscience 2019Quote: ... in the presence of the mGluR5 antagonist 2-methyl-6 (phenylethynyl)-pyridine (MPEP, 25 μM; Tocris Bioscience, Bristol, UK). Inhibitors were applied concomitantly from 30 min before to 30 min after DHPG/MPEP treatment ...
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bioRxiv - Neuroscience 2021Quote: ... The mGluR5 specific negative allosteric modulator MPEP hydrochloride (2-Methyl-6-(phenylethynyl)pyridine hydrochloride) was purchased from Tocris (1212) and administered to brain slices at 30 μM by bath perfusion ...
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bioRxiv - Neuroscience 2019Quote: ... N-[2-[[(Hexahydro-2-oxo-1H-azepin-3-yl)amino]carbonyl]phenyl]benzo[b]thiophene-2-carboxamide (ANA12, 10 µM) (Tocris), (9S,10R,12R)-2,3,9,10,11,12-Hexahydro-10-hydroxy-9-methyl-1-oxo-9,12-epoxy-1H-diindolo[1,2,3-fg:3’,2’,1’-kl]pyrrolo[3,4-i][1,6]benzodiazocine-10-carboxylic acid methyl ester (K252a ...
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bioRxiv - Immunology 2021Quote: ... and 2 ng/ml IL-2 (carrier-free; Tocris R&D Systems). Cells treated with only these functioned as the mock control ...
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bioRxiv - Neuroscience 2022Quote: ... or 20 μM 2-methylthyo-adenosine-5’-triphosphate (2-MeSATP, Tocris, 1062) over a 5-min period ...
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bioRxiv - Neuroscience 2024Quote: Commercially available (±)-7-hydroxy-DPAT HBr (Tocris; 50 mg, 0.15 mmol) was washed with saturated NaHCO3 aqueous solution and extracted with DCM ...
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bioRxiv - Systems Biology 2019Quote: ... 2μM IWP-2 (Tocris) and 10μM DAPT [goblet and enteroendocrine cells] (25).
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bioRxiv - Neuroscience 2021Quote: ... MLi-2 (Tocris #5756) was reconstituted in DMSO to a stock concentration of 10mM ...
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bioRxiv - Neuroscience 2022Quote: ... WIN55,212-2 (1038, Tocris), and Torin 2 (4248 ...
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bioRxiv - Cell Biology 2020Quote: ... MLi-2 (Tocris, 5756) was used at 1 µM ...
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bioRxiv - Pharmacology and Toxicology 2020Quote: WIN55,212-2 (Tocris, #1038), α-Humulene (Sigma Aldrich ...
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bioRxiv - Cell Biology 2020Quote: ... Torin-2 (Tocris 4248), rapamycin (CalBiochem 553211) ...
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bioRxiv - Cell Biology 2019Quote: ... and IWP-2 (Tocris) were added at 3µM and 1µM ...
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bioRxiv - Cell Biology 2023Quote: ... 2 µM Dorsomorphin (TOCRIS) and 2 µM XAV939 (Stemgent) ...
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bioRxiv - Developmental Biology 2023Quote: ... 2 µM CHIR99021 (Tocris) and 5µM Y27632 (Santa Cruz) ...
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bioRxiv - Physiology 2023Quote: ... 2 μM PD0332991 (Tocris), 10 ng/ml human BDNF (Miltenyi Biotec) ...
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bioRxiv - Cell Biology 2023Quote: ... 2 µM Dorsomorphin (Tocris), 10 µM SB-431542 (Tocris) ...
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bioRxiv - Neuroscience 2024Quote: ... DMH1 (2 μM, Tocris) and SB431542 (2 μM ...
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bioRxiv - Cancer Biology 2024Quote: ... AKTi-1/2 (Tocris), MK-2206 (VWR) ...
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bioRxiv - Cell Biology 2021Quote: 4-Methoxy-3-(2-phenylethoxy)-N,N-dipropylbenzeneethanamine hydrochloride (NE-100 hydrochloride) was purchased from Tocris (3133). Stock and work solutions were prepared using 100% dimethyl sulfoxide sterile-filtered (DMSO ...
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bioRxiv - Developmental Biology 2021Quote: ... early somite (1 day; 2 µM SB505124, 4 µM dorsomorphin, 500 nM PD173074 [cat. num. 3044; Tocris Bioscience ...
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Prelimbic proBDNF facilitates memory destabilization by regulation of neuronal function in juvenilesbioRxiv - Neuroscience 2022Quote: ... 3-(2-carboxypiperazin-4-yl)propyl-1-phosphonic acid (CPP; 32 ng/μL; Cat#01773, Tocris Bioscience), NVP-AAM077 (0.8 ng/μL ...
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Serotonin, Etonogestrel and breathing activity in murine Congenital Central Hypoventilation SyndromebioRxiv - Physiology 2022Quote: ... LP44 (4-[2-(methylthio)phenyl]-N-(1,2,3,4-tetrahydro-1-naphthalenyl)-1-piperazinehexanamide hydrochloride) was purchased from Tocris Bioscience (Bristol ...
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bioRxiv - Synthetic Biology 2022Quote: (5Z)-5[(3,5-Difluoro-4-hydroxyphenyl)methylene]-3,5-dihydro-2-methyl-3-(2,2,2-trifluoroethyl)-4H-imidazol-4-one (DFHBI-1T) was purchased from Tocris Bio-techne ...
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bioRxiv - Neuroscience 2020Quote: ... The following agents were used: L-(+)-2-amino-4-phophonobutyric acid (L-AP4; 20μM; Tocris Bioscience, catalog #0103), D-(-)-2-amino-5-phophonopentanoic acid (D-AP5 ...
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bioRxiv - Neuroscience 2020Quote: ... 2 μM CHIR99021 (Tocris Bioscience), 10 μM DAPT (Millipore Sigma) ...
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bioRxiv - Cell Biology 2022Quote: ... 2 μM dorsomorphin (Tocris, 3093) and 2 μM A-83 (Tocris ...
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bioRxiv - Developmental Biology 2021Quote: ... 2 µM forskolin (1099, Tocris), 200 nM phorbol-12 myristate-13 acetate (1201 ...
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bioRxiv - Cell Biology 2021Quote: ... and 2 μM DMH1 (Tocris) for 6 days ...
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bioRxiv - Neuroscience 2021Quote: ... 2-APB (Tocris, Cat.#: 1224), CPP (Tocris ...
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bioRxiv - Pharmacology and Toxicology 2020Quote: ... 2’Me-CCPA (Tocris, 2281), MRS1754 (Tocris ...
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bioRxiv - Cell Biology 2021Quote: ... Wnt inhibitor IWP-2(TOCRIS) and Srfp-2(R&D Systems ...
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bioRxiv - Cell Biology 2021Quote: ... MLi-2 (Tocris, cat #5756) was used at 1 μM in DMSO for 90 min ...
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bioRxiv - Neuroscience 2020Quote: ... 2 mg/ml biocytin (Tocris) was dissolved in the intracellular solution and cells were dialyzed for 20 minutes ...
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bioRxiv - Neuroscience 2020Quote: ... and 2-Aminoethoxydiphenylborane (1224, Tocris) in DMSO ...
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bioRxiv - Developmental Biology 2022Quote: ... 2 μM SU-5402 (Tocris), and 10 μM DAPT (Tocris) ...
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bioRxiv - Neuroscience 2022Quote: ... and Torin 2 (4248, Tocris). Other reagents used for making solutions were purchased from Sigma-Aldrich or Fisher Scientific.
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bioRxiv - Developmental Biology 2021Quote: ... SB-505124 (2 μM; Tocris) and FGF2 (20 ng/mL ...