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Citations for Tocris :
1 - 50 of 249 citations for 4 4 Fluorophenyl Ethynyl Phenyl Ethynyl Trimethylsilane since 2020
Citations are collected from bioRxiv only, the total number of publications could be much larger.
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bioRxiv - Neuroscience 2024Quote: ... VU0360172 [N-cyclobutyl-6-(2-(3-fluorophenyl)ethynyl) pyridine-3-carboxamide] was purchased from Tocris Bioscience (Bristol ...
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bioRxiv - Neuroscience 2021Quote: ... The mGluR5 specific negative allosteric modulator MTEP (3-((2-Methyl-1,3-thiazol-4-yl)ethynyl)pyridine hydrochloride) was purchased from Tocris (2921) and administered to brain slices at 1 μM by bath perfusion ...
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bioRxiv - Physiology 2024Quote: ... 4-(3-chloro-pyridin-2-yl)-piperazine-1-carboxylic acid (4-tert-butyl-phenyl)-amide (BCTC, Tocris #3875) 10 mM in DMSO ...
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bioRxiv - Physiology 2021Quote: ... resiniferatoxin and 4-(3-Chloro-2-pyridinyl)-N-[4-(1,1-dimethylethyl)phenyl]-1-piperazinecarboxamide (BCTC) were purchased from Tocris Bioscience or Adooq Bioscience and stock solutions were prepared in EtOH at 1 M and 100 mM ...
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bioRxiv - Immunology 2024Quote: ... The FFA2R antagonist CATPB ((S)-3-(2-(3-Chlorophenyl)acetamido)-4-(4-(trifluoromethyl) phenyl) butanoic acid) was from Tocris Bioscience (Bristol ...
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bioRxiv - Pharmacology and Toxicology 2023Quote: ... 2-[[6-amino-3,5-dicyano-4-[4-(cyclopropylmethoxy) phenyl]-2-pyridinyl]thio]-acetamide (BAY 60-6583; Tocris, 910487-58-0), 1-[2-chloro-6-[[(3-iodophenyl)methyl]amino]-9H-purin-9-yl]-1-deoxy-N-methyl-β-D-ribofuranuronamide (2-Chloro-IB-MECA ...
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bioRxiv - Neuroscience 2020Quote: ... 4-[(2S)-2-[(5-isoquinolinylsulfonyl)methylamino]-3-oxo-3-(4-phenyl-1-piperazinyl)propyl] phenyl isoquinolinesulfonic acid ester (KN-62; Tocris and HelloBio); D-AP5 (HelloBio) ...
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bioRxiv - Cell Biology 2022Quote: ... The FFA2R antagonist CATPB ((S)-3-(2-(3-chlorophenyl)acetamido)-4-(4-(trifluoromethyl)-phenyl) butanoic acid) was from Tocris (Britsol, UK).
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bioRxiv - Cancer Biology 2022Quote: ... the small molecule 3-[2-[(4-Fluorophenyl)methyl]imidazo[2,1-b]thiazol-6-yl]-2H-1-benzopyran-2-one (iMDK; TOCRIS Bio-techne, 9mg/kg), rapamycin (Sirolimus A8167 ...
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bioRxiv - Neuroscience 2024Quote: ... 7-Chloro-4-hydroxy-3-(3-phenoxy)phenyl-2(1H)-quinolinone (L-701-324; Tocris); (R)-3-(2-Carboxypiperazin-4-yl)propyl-1-phosphonic acid ((R)-CPP ...
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bioRxiv - Pharmacology and Toxicology 2023Quote: ... [2-Amino-4-[3-(trifluoromethyl)phenyl]-3-thienyl] phenylmethanone (VCP 171; Tocris, 1018830-99-3), 5-[2-(5-nitro-2-furanyl)ethenyl]-2-furancarboxylic acid ...
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Serotonin, Etonogestrel and breathing activity in murine Congenital Central Hypoventilation SyndromebioRxiv - Physiology 2022Quote: ... LP44 (4-[2-(methylthio)phenyl]-N-(1,2,3,4-tetrahydro-1-naphthalenyl)-1-piperazinehexanamide hydrochloride) was purchased from Tocris Bioscience (Bristol ...
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bioRxiv - Physiology 2022Quote: ... BPTU (1-(2-(2-(tert-butyl)phenoxy)pyridin-3-yl)-3-(4-(trifluoromethoxy) phenyl) urea was from Tocris Bioscience.
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bioRxiv - Neuroscience 2020Quote: The FPR2 agonist Compound-43 (N-(4-Chlorophenyl)-N-[2,3-dihydro-1-methyl-5-(1-methylethyl)-3-oxo-2-phenyl-1H-pyrazol-4-yl]-urea) and antagonist WRW4 (Trp-Arg-Trp-Trp-Trp-NH2) were purchased from Tocris Ltd ...
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bioRxiv - Neuroscience 2023Quote: ... and (3-chloro-4-fluoro-N-[(4-([2-(phenylcarbonyl)hydrazino]carbonyl) phenyl)methyl]benzene-sulfonamide) (TCN-201) (Hansen et al., 2012)were obtained from Tocris Bioscience ...
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bioRxiv - Cell Biology 2024Quote: ... and P2Y1 antagonist 1-(2- (2- tert-butylphenoxy)pyridin-3-yl)-3-(4-(trifluoromethoxy)phenyl)urea (BPTU; BMS- 646786, #870544-59-5) were obtained from Tocris Bioscience (Bristol ...
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bioRxiv - Developmental Biology 2022Quote: 4-Hydroxytamoxifen (4-OHT) (Tocris Bioscience) was dissolved in corn oil (Millipore-Sigma ...
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bioRxiv - Neuroscience 2020Quote: ... 4-aminopyrimidine (4-ap, 30 µM, Tocris) and/or Tetrodotoxin (TTX ...
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bioRxiv - Neuroscience 2020Quote: ... 100 4-aminopyridine (4-AP) (Tocris Bioscience). To determine possible changes in intrinsic excitability ...
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bioRxiv - Biophysics 2022Quote: ... or 4 μM GsMTx-4 (Tocris 4912) were incubated for 15 min ...
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bioRxiv - Neuroscience 2023Quote: ... 100 μM 4-aminopyridin (4-AP, Tocris) and 20 mM tetraethylammonium chloride (TEA ...
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bioRxiv - Neuroscience 2020Quote: ... or 4-aminopyridine (4-AP, Cat. No. 0940, Tocris), diluted in culture medium at a final concentration of 1 μM and 50 μM ...
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bioRxiv - Neuroscience 2023Quote: ... 4-Aminopyridine (4- AP; 100 µM; Tocris, Item# 0940), 6,7-Dinitroquinoxaline-2,3-dione (DNQX ...
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bioRxiv - Cell Biology 2022Quote: ... 1,1-Dimethyl-4-diphenylacetoxypiperidinium iodide (4-DAMP, 0.1 µM, Tocris), U73122 (10 µM ...
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bioRxiv - Neuroscience 2022Quote: ... Exendin-4 (Tocris) was administered at 0.004 to 0.04 mg/kg ...
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bioRxiv - Neuroscience 2022Quote: ... DSP-4 (Tocris) was dissolved in saline and a single dose (75 mg/kg BW ...
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bioRxiv - Neuroscience 2024Quote: DSP-4 (Tocris) was dissolved in saline ...
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bioRxiv - Cell Biology 2021Quote: ... interleukin-1 receptor-associated kinase 1 and 4 (IRAK 1/4; IRAK 1/4 inhibitor, 0.1 μM; Tocris); TANK-binding kinase 1 (TBK1 ...
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bioRxiv - Neuroscience 2024Quote: ... Kv1-4 Channels were blocked with 4-aminopyridine (1 mM, Tocris), Kv7 channels with XE991 dihydrochloride (20 µM ...
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bioRxiv - Cancer Biology 2022Quote: ... and 1,3-Bis(4-hydroxyphenyl)-4-methyl-5-[4-(2-piperidinylethoxy)phenol]-1H-pyrazoledihydro-chloride (MPP; cat# 1991) were purchased from Tocris Bioscience ...
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bioRxiv - Neuroscience 2021Quote: ... The following chemical reagents were used: 4-aminopyridine (4-AP, TOCRIS, #940), ADX 71743 (TOCRIS ...
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bioRxiv - Neuroscience 2021Quote: ... 4-AP (Tocris, UK) was stored as a stock solution of 100 mM in ACSF at -20°C and applied to the bath at 5 mM ...
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bioRxiv - Developmental Biology 2021Quote: ... CHIR99021 (4 μM; Tocris), FGF2 (20 ng/mL ...
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bioRxiv - Cell Biology 2023Quote: ... 4-IPP (Tocris, 3429), and Brefeldin A (Millipore-Sigma ...
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bioRxiv - Genetics 2024Quote: ... 4 μM CHIR99021 (Tocris), 20 ng/mL FGF2 (PeproTech ...
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bioRxiv - Neuroscience 2024Quote: ... 4-DAMP (10μM, Tocris) and vehicle (DMSO ...
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bioRxiv - Cell Biology 2024Quote: ... 4 μM CHIR99021 (Tocris), 20 ng/mL FGF2 (PeproTech ...
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bioRxiv - Physiology 2021Quote: ... L-364,373 (R-L3 or 5-(2-Fluorophenyl)-1,3-dihydro-3-(1H-indol-3-ylmethyl)-1-methyl-2H-1,4-benzodiazepin-2-one) (Tocris Cookson; Bristol, UK) and mefenamic (dimethylphenylaminobenzoic ...
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bioRxiv - Cell Biology 2020Quote: ... 2-(4-chlorophenyl)-3-methyl-N-(thiazole-2-yl)butanamide (4-CMTB; Tocris) was used as a FFAR2-specific agonist and AR420626 (Cayman ...
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bioRxiv - Neuroscience 2023Quote: ... in combination with potassium channel blocker 4-aminopyridine (4-AP, 1 mM, Tocris) to facilitate transmitter release at monosynaptic connections from RSC to ChC and recorded the PSP amplitudes (Figure 1H) ...
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bioRxiv - Bioengineering 2021Quote: ... Photoinitiator lithium phenyl-2,4,6-trimethylbenzoylphosphinate (LAP) (Tocris, 6146) at concentrations of 0.1% ...
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bioRxiv - Cancer Biology 2024Quote: To induce the degradation of AID-NCL, cells were treated with 5-phenyl-indole-3-acetic acid (phenyl-auxin, 5-Ph-IAA) (Tocris, #7392). To block the interaction between APC/C and cdc20 ...
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bioRxiv - Neuroscience 2021Quote: ... 4-DAMP (Catalog #0482, Tocris), AFDX-384 (Catalog #1345 ...
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bioRxiv - Cancer Biology 2021Quote: ... 4 μM IWP-2 (Tocris), and 1 μM A83-01 (Tocris) ...
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bioRxiv - Cell Biology 2020Quote: ... KN-62 (4 μM, TOCRIS), BAPTA-AM (10 μM ...
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bioRxiv - Neuroscience 2021Quote: ... 4 µM SR 95531 (Tocris) and 10 µM DL-AP5 (Tocris) ...
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bioRxiv - Developmental Biology 2020Quote: ... 4 μM IWP-2 (Tocris), and 1 μM A83-01 (Tocris ...
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bioRxiv - Neuroscience 2023Quote: ... Topiramate (Tocris, #97240-79-4), and Carbamazepine (Tocris ...
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bioRxiv - Neuroscience 2023Quote: ... and 4 μM XAV (Tocris). On DIV 04 ...
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bioRxiv - Neuroscience 2024Quote: ... or 4-DAMP (10μM, Tocris) was added and incubated for a further 24h ...