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Citations for Tocris :
401 - 450 of 976 citations for 6 Propyl 2 thioxo 2 3 dihydropyrimidin 4 1H one since 2019
Citations are collected from bioRxiv only, the total number of publications could be much larger.
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bioRxiv - Neuroscience 2021Quote: We inhibited LRRK2 kinase activity with the selective LRRK2 inhibitor MLi-2 (Tocris 5756). MLi-2 has low solubility in water ...
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bioRxiv - Genomics 2021Quote: ... followed by 2 uM of the Wnt signaling inhibitor Wnt-C59 (5148, Tocris Bioscience). Cells start to spontaneously beat between days 7-10 ...
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bioRxiv - Neuroscience 2022Quote: ... and L-2-amino-5-phosphonopentanoic acid (APV, an NMDA receptor blocker) from Tocris. APV ...
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bioRxiv - Neuroscience 2023Quote: ... and 50 μM 2-amino-5-phosphonopentanoic acid (D-AP5; Tocris Bioscience, Cambridge, UK) to avoid spontaneous network activation ...
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bioRxiv - Neuroscience 2022Quote: ... and 50 μM D,L-2-amino-5-phosphonovaleric acid (AP5, TOCRIS bioscience #0105). NH4Cl perfusions were done with 50 mM NH4Cl in substitution of 50 mM NaCl (pH 7.4) ...
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bioRxiv - Developmental Biology 2021Quote: ... CHIR99021 (6 μM; Tocris), FGF2 (20 ng/mL ...
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bioRxiv - Neuroscience 2020Quote: ... 4-Butoxy-N-[1,4-dihydro-2-(4-methoxyphenyl)-4-oxo-3(2H)-quinazolinyl]benzamide) and antagonist WRW4 (Trp-Arg-Trp-Trp-Trp-Trp-NH2) were purchased from Tocris Ltd ...
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bioRxiv - Neuroscience 2019Quote: ... (+)-4-[(αR)-α-((2S,5R)-4-Allyl-2,5-dimethyl-1-piperazinyl)-3-methoxybenzyl]-N,N-diethylbenzamide (SNC 80) (20mg/kg; Tocris) dissolved in 1mM HCl in saline.
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bioRxiv - Pharmacology and Toxicology 2019Quote: ... or 2 mM (R,S)-3,5-DHPG (mGlu1/5 agonist, Tocris 0805 and 0342 respectively), and the astrocyte marker Sulforhodamine 101 (40 μM ...
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bioRxiv - Neuroscience 2020Quote: ... Animals were then immobilized by immersion in a solution of 2 mM pancurionium dibromide (Tocris) in 0.1X MBSH for 2-5 min ...
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bioRxiv - Neuroscience 2019Quote: ... The exogenous DREADD ligand clozapine-N-oxide CNO (2 mg/kg) was purchased from Tocris Bioscience (Bristol ...
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bioRxiv - Neuroscience 2021Quote: ... 1,2-bis(2-aminophenoxy)ethane-N,N,N’,N’-tetraacetic acid (BAPTA, 50 µM, Tocris); and 1,2-Bis(2-aminophenoxy)ethane-N,N,N’,N’-tetra-acetic acid tetrakis (acetoxymethylester ...
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bioRxiv - Neuroscience 2021Quote: ... 25 μM of d-(-)-2-amino-5-phosphonopentanoic acid (D-AP5, 0106, Tocris Bioscience, UK), and 10 μM of SR95531 (SR ...
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bioRxiv - Cell Biology 2021Quote: ... and human vasopressin type 2 receptor (V2R) with [Arg8]-vasopressin (AVP; Tocris 2935, in water). The transfected β-arrestins are of bovine origin ...
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bioRxiv - Neuroscience 2019Quote: ... D-2-amino-5-phosphonovalerate (“D-AP5”, 50 mM in PBS, Tocris Cat No 0106); Retigabine (100 mM in DMSO ...
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bioRxiv - Genomics 2020Quote: ... supplemented with SMAD inhibitors (DMH-1 2 μM Tocris, Cat.: #4423; SB431542-10 μM Tocris, Cat. ...
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bioRxiv - Genomics 2021Quote: ... 1 µM DMH1-HCl (in house synthesized, Vanderbilt University) and 240 nM IWP-2 (Tocris). On day 8 of differentiation ...
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bioRxiv - Biochemistry 2022Quote: ... and E3 ligase recruiter building blocks thalidomide - linker 2 (#6468/25) were purchased from Tocris Bioscience (Minneapolis ...
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bioRxiv - Neuroscience 2023Quote: ... and exposure to a cocktail of small molecules containing 2 μM each of Dorsomorphin (Tocris), A83-01 (Tocris ...
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The CB1 receptor interacts with cereblon and drives cereblon deficiency-associated memory shortfallsbioRxiv - Neuroscience 2023Quote: ... a single submaximal concentration (10 µM) of WIN-55,212-2 or HU-210 (Tocris #0966) was used ...
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bioRxiv - Neuroscience 2023Quote: ... organoids were placed in HEPES buffer containing CNQX/APV (2 µM/50 µM, Tocris Bioscience) and imaged immediately.
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bioRxiv - Genomics 2023Quote: ... spent media was replaced with fresh CDM containing 2 µM Wnt-C59 (5148, Tocris Bioscience). CDM was used to replace media on Days 5 ...
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HOIL-1L deficiency induces cell cycle alteration which causes immaturity of myocyte and fibrogenesisbioRxiv - Cell Biology 2023Quote: ... the medium was replaced with differentiation medium containing 5 μM IWP-2 (TOCRIS, Cat.# 3533), a Wnt inhibitor ...
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bioRxiv - Neuroscience 2024Quote: ... USA) and superfused with ACSF containing 2 mM CaCl2 and 20 µM bicuculline methiodide (Tocris) at a rate of 3 – 4 ml/min at RT ...
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bioRxiv - Neuroscience 2022Quote: ... 12-well plates at 3-4 × 105 cells/well in mTeSR1 with 10 µM rho-kinase inhibitor (Y-27632; Tocris, 1254). Medium without the inhibitor was replaced daily until the cells reach 80-100% confluency ...
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bioRxiv - Biochemistry 2022Quote: ... Positive clones were analyzed by Sanger sequencing with primers #3 and #4 (Integrated DNA Technologies, Supplementary Table S5) and degradation upon dTAG-13 (Tocris, 6605) treatment was confirmed by Western Blot by a-Chaf1a antibody (65) ...
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bioRxiv - Neuroscience 2022Quote: ... and PACAP(6-38) (Tocris). For high K+ stimulation ...
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bioRxiv - Neuroscience 2022Quote: ... and 6-OHDA (2547, Tocris) were injected into the left hemisphere of substantia nigra pars compacta (SNpc ...
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bioRxiv - Neuroscience 2023Quote: ... 6-OHDA hydrobromide (Tocris Bioscience) was dissolved in ice-cold 0.02% ascorbic acid dissolved in saline to a concentration of 4 μg/μl ...
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bioRxiv - Cell Biology 2024Quote: ... bEnd.3 cells were treated with either 3-methyladenine (3-MA, #1292 Tocris, MN, USA) or rapamycin (Rapa ...
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bioRxiv - Neuroscience 2020Quote: ... WIN 55,212-2 (WIN, 0.5 µg/0.5-µL infusion/hemisphere; n = 11; Tocris Bioscience, Minneapolis, MN) or VEH (10% DMSO ...
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bioRxiv - Cancer Biology 2022Quote: ... 2% Sodium deoxycholate and 0.2% SDS including protease inhibitors (Aprotinin (TOCRIS Bioscience Cat. no. 4139/10) Leupeptin (Fisher Scientific ...
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bioRxiv - Genomics 2019Quote: ... the previously described medium was replaced with heart medium containing 2 μM Wnt-C59 (Tocris, 5148). On days 5 ...
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bioRxiv - Developmental Biology 2021Quote: ... Lin- c-Kit+ cells were sorted into 2%FCS-PBS with 100µM IWR-1 (Tocris, 3532) or control vehicle ...
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bioRxiv - Microbiology 2020Quote: ... cells were pretreated for 3h before infection with Tautomycetin (0.8 μM, Tocris Bioscience, 119757-73-2) or Okadaic acid (0.1 μM ...
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bioRxiv - Molecular Biology 2021Quote: Cells were treated for 2 hrs with vehicle (DMSO) or with 250 nM Torin1 (Tocris Biosciences), or for 1 hr with 50 μM Ly29004 (Tocris Biosciences ...
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bioRxiv - Neuroscience 2022Quote: ... we slowly infused 200 nl of the GABAA receptor agonist muscimol (Tocris; 2 μM in saline) into the target area using a micro-syringe pump (KD Scientific ...
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bioRxiv - Neuroscience 2022Quote: The β3AR-selective antagonist SR59230A (2 mg/kg/day or 10 mg/kg/day; Tocris Bioscience) or vehicle (2:3 ratio of DMSO:0.9% saline ...
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bioRxiv - Biochemistry 2023Quote: ... Cannabinoid ligands (anandamide [AEA], 2-arachydonyl-glycerol [2AG], SR144528, HU210, HU308, cannabinol) were obtained from Tocris Bioscience and dissolved in DMSO to a storage concentration of 10 mM ...
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bioRxiv - Developmental Biology 2023Quote: ... at a density of 2 × 103 cells/cm2 with 10µM ROCK inhibitor (Y-27632; Tocris, 1254) added in culture medium for 1 day after hESCs passaging ...
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bioRxiv - Cell Biology 2024Quote: ... the WNT signaling inhibitor IWP-2 (2μM in DMSO, day 21-42, Tocris Bioscience, Bristol, UK), the hedgehog inhibitor cyclopamine (10μM in DMSO ...
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bioRxiv - Developmental Biology 2024Quote: ... Cells were treated as control or with 2 µM DDR1 inhibitor DDR1-in-1 (Tocris 5077) or 5 µM RUNX1 inhibitor AI-10-104 (Aobious AOB17076) ...
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bioRxiv - Developmental Biology 2022Quote: 4-Hydroxytamoxifen (4-OHT) (Tocris Bioscience) was dissolved in corn oil (Millipore-Sigma ...
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bioRxiv - Neuroscience 2020Quote: ... co-applied with the competitive α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid AMPA/kainate receptor antagonist CNQX (Tocris; 20 μM) (n=13) ...
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bioRxiv - Neuroscience 2020Quote: ... 4-aminopyrimidine (4-ap, 30 µM, Tocris) and/or Tetrodotoxin (TTX ...
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bioRxiv - Neuroscience 2020Quote: ... 100 4-aminopyridine (4-AP) (Tocris Bioscience). To determine possible changes in intrinsic excitability ...
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bioRxiv - Biophysics 2022Quote: ... or 4 μM GsMTx-4 (Tocris 4912) were incubated for 15 min ...
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bioRxiv - Neuroscience 2023Quote: ... 100 μM 4-aminopyridin (4-AP, Tocris) and 20 mM tetraethylammonium chloride (TEA ...
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bioRxiv - Neuroscience 2020Quote: ... 250 nM PACAP 6-38 (Tocris), 20 µM Bicuculline (Cayman chemical) ...
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bioRxiv - Neuroscience 2019Quote: ... 6-OHDA (Tocris; conjugated with HBr) was injected bilaterally in a 4 × 3 grid at AP coordinates 5.1 ...