Labshake search
Citations for Tocris :
201 - 250 of 1132 citations for 6 Bromo 2 trifluoromethyl 3H imidazo 4 5 b pyridine since 2019
Citations are collected from bioRxiv only, the total number of publications could be much larger.
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bioRxiv - Neuroscience 2020Quote: The FPR2 agonist Compound-43 (N-(4-Chlorophenyl)-N-[2,3-dihydro-1-methyl-5-(1-methylethyl)-3-oxo-2-phenyl-1H-pyrazol-4-yl]-urea) and antagonist WRW4 (Trp-Arg-Trp-Trp-Trp-NH2) were purchased from Tocris Ltd ...
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bioRxiv - Microbiology 2022Quote: ... 3 μl of 10 mM of NBD-(linezolid-7-nitrobenz-2-oxa-1,3-diazol-4-yl)-amino-D-alanine (NADA) (Tocris Bioscience) was added to the resuspension ...
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bioRxiv - Neuroscience 2023Quote: ... and (3-chloro-4-fluoro-N-[(4-([2-(phenylcarbonyl)hydrazino]carbonyl) phenyl)methyl]benzene-sulfonamide) (TCN-201) (Hansen et al., 2012)were obtained from Tocris Bioscience ...
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bioRxiv - Neuroscience 2019Quote: ... and 20 mM 4-aminopyridine (4-AP; Tocris) were included for more stringent isolation of monosynaptic transmission (Cruikshank et al. ...
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bioRxiv - Neuroscience 2021Quote: ... d-2-Amino-5-phosphonovaleric acid (d-AP5, 50µM) and the sodium (Na+) channel blocker tetrodotoxin (TTX, 1 µM Tocris). Individual traces (5 sec duration ...
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bioRxiv - Neuroscience 2019Quote: ... To block NMDA receptors we used D- (-)-2-Amino-5-phosphonopentanoic acid (D-AP5, Tocris, 10 μM final concentration). To block glycinergic inhibition ...
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bioRxiv - Biochemistry 2020Quote: ... 4-[(2-Butyl-6,7-dichloro-2-cyclopentyl-2,3-dihydro-1-oxo-1H-inden-5-yl)oxy] butanoic acid (DCPIB) was purchased from Tocris Bioscience and reconstituted to 50 mM in DMSO ...
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bioRxiv - Neuroscience 2020Quote: ... 20 μM 6,7-dinitroquinoxaline-2,3-dione (DNQX) and 20 μM D-(-)-2-amino-5-phosphopentanoic acid (D-AP5) (Tocris Bioscience) to block glycine- ...
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bioRxiv - Cell Biology 2021Quote: ... AKT (20 μM MK2206, Cayman Biochemicals #1032350-13-2) and myosin ATPase activity inhibitor (5 μM Blebbistatin, Tocris #1852).
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bioRxiv - Immunology 2020Quote: ... 4-[(2-Butyl-6,7-dichloro-2-cyclopentyl-2,3-dihydro-1-oxo-1H-inden-5-yl)oxy]butanoic acid (DCPIB, 1540) was from Tocris. NS3728 and NBC19 were made at the University of Manchester.
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bioRxiv - Neuroscience 2019Quote: ... and the monoamine oxidase A & B inhibitor bifemelane (50 µM; Tocris).
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bioRxiv - Immunology 2020Quote: ... B cells were incubated with FFN200 (10μM, Tocris, catalogue number: 5911), a selective substrate for the vesicular monoamine transporter-2 for 1.15h ...
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bioRxiv - Cancer Biology 2023Quote: ... 500 nM TGF-b type I receptor inhibitor A83-01 (Tocris), 10 µM P38 inhibitor SB202190 (Sigma-Aldrich) ...
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bioRxiv - Cancer Biology 2020Quote: ... 6-Bnz-cAMP was purchased from Tocris Bioscience (5255) ...
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bioRxiv - Neuroscience 2020Quote: ... 6-OHDA(100 mg/kg, Tocris, UK) was given every 2 d ...
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bioRxiv - Cell Biology 2022Quote: ... 3 µM or 6 µM proTAME (Tocris) and mounted in modified rose chambers ...
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bioRxiv - Cell Biology 2022Quote: ... 3 µM or 6 µM proTAME (Tocris). For monastrol arrest and release experiments ...
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bioRxiv - Cell Biology 2022Quote: ... 3 µM or 6 µM proTAME (Tocris).
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bioRxiv - Cell Biology 2022Quote: ... 6 µM or 20 µM proTAME (Tocris) or 2 µM UMK57 or UMK95 during imaging ...
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bioRxiv - Cell Biology 2023Quote: ... RAC1 inhibitor (CAS1177865-17-6; Tocris Biosciences) was used at 100 µM ...
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bioRxiv - Neuroscience 2020Quote: ... co-applied with the competitive α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid AMPA/kainate receptor antagonist CNQX (Tocris; 20 μM) (n=13) ...
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bioRxiv - Neuroscience 2023Quote: ... Drug treatments correspond to a single dose of cocaine hydrochloride at 20 mg/kg (Medisca, cat# 53-21-4, Canada) or D-amphetamine sulfate at 5 mg/kg (Tocris, 2813, UK) at doses known to increase locomotion87 ...
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bioRxiv - Biochemistry 2024Quote: ... The filtrate was diluted two times the volume with buffer UA (8 M urea [Acros Organics, CAS No. 57-13-6], 50 mM sodium acetate [Tocris CAS No. 127-09-3], pH 4). This was loaded onto a HiPrep SP HP 16/10 (Cytiva ...
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bioRxiv - Neuroscience 2020Quote: ... or 4-aminopyridine (4-AP, Cat. No. 0940, Tocris), diluted in culture medium at a final concentration of 1 μM and 50 μM ...
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bioRxiv - Neuroscience 2023Quote: ... 4-Aminopyridine (4- AP; 100 µM; Tocris, Item# 0940), 6,7-Dinitroquinoxaline-2,3-dione (DNQX ...
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bioRxiv - Developmental Biology 2019Quote: ... From day 2 to day 4 the medium was additionally supplemented with BMP and TGFβ inhibitors (Noggin, Peprotech and SB431542, Tocris Bioscience). Treatment with MEK inhibitor (PD184352 ...
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bioRxiv - Neuroscience 2021Quote: ... Four of the rats were also infused with 2 μL of either physiological saline or 5 μg/μL yohimbine (Tocris) with a flow rate of 0.5 μL/min as previously reported (Caetano et al. ...
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bioRxiv - Neuroscience 2020Quote: ... QX-314 (Cat No. 1014); and D-2-amino-5-phosphonovalerate (D-AP5; Cat No. 0106) were purchased from Tocris.
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A Bidirectional Switch in the Shank3 Phosphorylation State Biases Synapses toward Up or Down ScalingbioRxiv - Neuroscience 2021Quote: ... 6 hrs (Figure 6 – figure supplement 2) or 24 hrs after transfection (the remaining experiments) neurons were treated with tetrodotoxin (TTX, 5 µM, Tocris) for ∼16 hours ...
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bioRxiv - Neuroscience 2020Quote: ... During BQA experiments the ACSF solution contained the following substances: 10 μM D-(−)-2-Amino-5-phosphonopentanoic acid (D-AP5) (Tocris), 10 μM 2,3-Dioxo-6-nitro-1,2,3,4-tetrahydrobenzo[f]quinoxaline-7-sulfonamide (NBQX ...
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bioRxiv - Microbiology 2023Quote: ... cells were resuspended in 25 µl PBS together with 0.25 µl of 5 mM 3-[[(7-Hydroxy-2-oxo-2H-1-benzopyran-3-yl) carbonyl]amino]-D-alanine hydrocholoride (HADA) (Tocris) dissolved in DMSO ...
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bioRxiv - Neuroscience 2022Quote: ... Animals were subsequently transferred to 1.5mL Lo-Bind tube and treated with 6-hydroxydopamine (6-OHDA; Tocris, Bristol, UK) containing 2mM ascorbic acid for one-hour ...
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bioRxiv - Cancer Biology 2021Quote: ... 0.5 μM TGF-b type I receptor inhibitor A83-01 (Tocris Bioscience) and 1μM PGE2 (Tocris Bioscience) ...
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bioRxiv - Cancer Biology 2021Quote: ... 5000 nM TGF-b type I receptor inhibitor A83-01 (Tocris #2939), 10 nM Prostaglandin E2 (Tocris #2296) ...
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bioRxiv - Neuroscience 2023Quote: ... 7-(Hydroxyimino)cyclopropa[b]chromen-1a-carboxylate ethyl ester (CPCCOEt, Tocris®); Tetrodotoxin (TTX ...
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Nucleocytoplasmic transport rates are regulated by cellular processes that modulate GTP availabilitybioRxiv - Cell Biology 2023Quote: Cells were treated with cytochalasin B (Tocris Biosciences, 20 µM, 10 min) and latrunculin B (MilliporeSigma ...
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bioRxiv - Cell Biology 2022Quote: ... 1,1-Dimethyl-4-diphenylacetoxypiperidinium iodide (4-DAMP, 0.1 µM, Tocris), U73122 (10 µM ...
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bioRxiv - Neuroscience 2021Quote: ... NMDA receptor (R) dependency was tested by application of an NMDAR antagonist (APV 50 µM, DL-2-Amino-5-phosphonopentanoic acid, Tocris, Germany) in the bath solution ...
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bioRxiv - Pharmacology and Toxicology 2020Quote: ... and a fourth group (DZP) received 2 mg/kg diazepam (CAS #439-14-5; Tocris, 2805; German-Ponciano et al., 2020) as a pharmacological control of anxiolytic activity ...
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bioRxiv - Physiology 2021Quote: ... Picrotoxin (100 µM) was used to block GABAA-receptor-mediated currents and D-2-amino-5-phosphonovalerate (APV; 20 µMm, Tocris Bioscience), and 6-cyano-7-nitroquinoxaline-2,3-dione (CNQX ...
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bioRxiv - Neuroscience 2022Quote: ... containing 10 μM 6-cyano-7-nitroquinoxaline-2,3-dione (CNQX) and 50 μM D,L-2-amino-5-phosphonovaleric acid (AP5) (both from Tocris, Bristol, UK) to block recurrent glutamatergic signaling.
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bioRxiv - Neuroscience 2023Quote: ... The following compounds were added to raCSF as indicated in the Results section: D-(-)-2-Amino-5-phosphonopentanoic acid (D-APV, 100 μM dissolved in H2O; Tocris Bioscience), (5S,10R)-(+)-5-Methyl-10,11-dihydro-5H-dibenzo[a,d] cyclohepten-5,10-imine maleate (MK-801 ...
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bioRxiv - Neuroscience 2024Quote: ... Both control and CACNA1A+/− networks at DIV49 were treated acutely with 100 µM D-2-amino-5-phosphonovalerate (D-AP5; Tocris, #0106) for 60 min ...
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bioRxiv - Biophysics 2021Quote: ... Cells were treated with 6 μM CHIR99021 (Tocris) for 48 hours on day 0 ...
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bioRxiv - Developmental Biology 2021Quote: ... 6 μM Chir 99021 (Tocris cat. no. 4423), 20ng/ml murine bFGF (PeproTech cat ...
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bioRxiv - Neuroscience 2020Quote: ... GABAA (6 µM bicuculline metiodide, Tocris, Bristol, UK) or GABAB (100 µM CGP46381 ...
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bioRxiv - Neuroscience 2020Quote: ... and Pyridone 6 (#6577) were purchased from Tocris Bioscience (Bristol ...
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bioRxiv - Neuroscience 2020Quote: ... 6-cyano-7-nitroquinoxaline-2,3-dione (CNQX, Tocris), 2,3-dihydroxy-6-nitro-7-sulfamoyl-benzo[f]quinoxaline-2,3-dione (NBQX ...
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bioRxiv - Molecular Biology 2020Quote: ... KN-62 and Inca-6 were from Tocris Bioscience (Minneapolis ...
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bioRxiv - Pharmacology and Toxicology 2021Quote: ... and SN-6 (2184) were purchased from Tocris, UK ...