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Citations for Tocris :
601 - 650 of 1908 citations for 6H Pyrazolo 3 4 b pyridin 6 one 3 cyclobutyl 1 2 4 5 tetrahydro 4 methyl 9CI since 2019
Citations are collected from bioRxiv only, the total number of publications could be much larger.
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bioRxiv - Neuroscience 2020Quote: ... 20 μM 6,7-dinitroquinoxaline-2,3-dione (DNQX) and 20 μM D-(-)-2-amino-5-phosphopentanoic acid (D-AP5) (Tocris Bioscience) to block glycine- ...
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bioRxiv - Cell Biology 2021Quote: ... AKT (20 μM MK2206, Cayman Biochemicals #1032350-13-2) and myosin ATPase activity inhibitor (5 μM Blebbistatin, Tocris #1852).
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bioRxiv - Physiology 2023Quote: ... animals either received vehicle (1 µl DMSO; n = 6) or the DREADD ligand clozapine n-oxide (CNO, Tocris; 0.1 mg/µl DMSO ...
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bioRxiv - Neuroscience 2019Quote: ... and the monoamine oxidase A & B inhibitor bifemelane (50 µM; Tocris).
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bioRxiv - Immunology 2020Quote: ... B cells were incubated with FFN200 (10μM, Tocris, catalogue number: 5911), a selective substrate for the vesicular monoamine transporter-2 for 1.15h ...
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bioRxiv - Cancer Biology 2023Quote: ... 500 nM TGF-b type I receptor inhibitor A83-01 (Tocris), 10 µM P38 inhibitor SB202190 (Sigma-Aldrich) ...
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bioRxiv - Neuroscience 2020Quote: ... we injected one of two doses of synthetic oxytocin (Tocris) into the BNSTam of females and males naïve to stress ...
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bioRxiv - Cancer Biology 2020Quote: ... 6-Bnz-cAMP was purchased from Tocris Bioscience (5255) ...
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bioRxiv - Neuroscience 2020Quote: ... 6-OHDA(100 mg/kg, Tocris, UK) was given every 2 d ...
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bioRxiv - Cell Biology 2022Quote: ... 6 µM or 20 µM proTAME (Tocris) or 2 µM UMK57 or UMK95 during imaging ...
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bioRxiv - Cell Biology 2023Quote: ... RAC1 inhibitor (CAS1177865-17-6; Tocris Biosciences) was used at 100 µM ...
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bioRxiv - Cell Biology 2022Quote: The mitogen-activated protein kinase kinase 1/2 (MEK1/2) inhibitor U0126 and the p38 MAPK inhibitor SB203580 were purchased from Tocris Bioscience (Bristol ...
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bioRxiv - Neuroscience 2023Quote: ... The [11C]MeOTf was slowly bubbled into a reaction vial containing 0.2mg 11-(1-Piperazinyl)-5H-dibenzo[b,e][1,4]diazepine precursor (Tocris, Bio-Techne Corp., Minneapolis, MN) and 0.3mL anhydrous MeCN (ThermoFisher Scientific ...
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bioRxiv - Cell Biology 2021Quote: ... 1 volume of phase separation buffer containing 5 μM A-485 (Tocris, 6387) was added and the mixture incubated for 10 min at room temperature before transferring the suspension to a passivated 384-well microscopy plate well.
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bioRxiv - Neuroscience 2022Quote: ... a stable baseline was established for 5 min and 1 μM oxytocin (Tocris) in ACSF was washed on for 30 min ...
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bioRxiv - Neuroscience 2023Quote: ... 5 mM HEPES and 30 mM Glucose) with 1 µM tetrodotoxin (TTX) (Tocris) for 30 s ...
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bioRxiv - Neuroscience 2021Quote: ... Four of the rats were also infused with 2 μL of either physiological saline or 5 μg/μL yohimbine (Tocris) with a flow rate of 0.5 μL/min as previously reported (Caetano et al. ...
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bioRxiv - Neuroscience 2020Quote: ... QX-314 (Cat No. 1014); and D-2-amino-5-phosphonovalerate (D-AP5; Cat No. 0106) were purchased from Tocris.
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A Bidirectional Switch in the Shank3 Phosphorylation State Biases Synapses toward Up or Down ScalingbioRxiv - Neuroscience 2021Quote: ... 6 hrs (Figure 6 – figure supplement 2) or 24 hrs after transfection (the remaining experiments) neurons were treated with tetrodotoxin (TTX, 5 µM, Tocris) for ∼16 hours ...
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bioRxiv - Neuroscience 2020Quote: ... During BQA experiments the ACSF solution contained the following substances: 10 μM D-(−)-2-Amino-5-phosphonopentanoic acid (D-AP5) (Tocris), 10 μM 2,3-Dioxo-6-nitro-1,2,3,4-tetrahydrobenzo[f]quinoxaline-7-sulfonamide (NBQX ...
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bioRxiv - Neuroscience 2020Quote: ... and re-plated at 1:6 ratio on Matrigel-coated plate in neural medium supplemented with 1μM CHIR99021 (Tocris), 2μM DMH1 (Tocris) ...
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bioRxiv - Neuroscience 2020Quote: ... and re-plated at 1:6 ratio on Matrigel-coated plate in neural medium supplemented with 3μM CHIR99021 (Tocris), 2μM DMH1 (Tocris) ...
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bioRxiv - Neuroscience 2022Quote: ... Animals were subsequently transferred to 1.5mL Lo-Bind tube and treated with 6-hydroxydopamine (6-OHDA; Tocris, Bristol, UK) containing 2mM ascorbic acid for one-hour ...
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bioRxiv - Physiology 2023Quote: Mice of 20 weeks of aged were injected retro-orbitally with 10 mM L-NMMA (NG-methyl-L-arginine acetate salt, Tocris Bioscience, 0771) to reach a final systemic concentration of 10 µM ...
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bioRxiv - Cancer Biology 2021Quote: ... 0.5 μM TGF-b type I receptor inhibitor A83-01 (Tocris Bioscience) and 1μM PGE2 (Tocris Bioscience) ...
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bioRxiv - Cancer Biology 2021Quote: ... 5000 nM TGF-b type I receptor inhibitor A83-01 (Tocris #2939), 10 nM Prostaglandin E2 (Tocris #2296) ...
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bioRxiv - Neuroscience 2023Quote: ... 7-(Hydroxyimino)cyclopropa[b]chromen-1a-carboxylate ethyl ester (CPCCOEt, Tocris®); Tetrodotoxin (TTX ...
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Nucleocytoplasmic transport rates are regulated by cellular processes that modulate GTP availabilitybioRxiv - Cell Biology 2023Quote: Cells were treated with cytochalasin B (Tocris Biosciences, 20 µM, 10 min) and latrunculin B (MilliporeSigma ...
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bioRxiv - Neuroscience 2021Quote: ... NMDA receptor (R) dependency was tested by application of an NMDAR antagonist (APV 50 µM, DL-2-Amino-5-phosphonopentanoic acid, Tocris, Germany) in the bath solution ...
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bioRxiv - Pharmacology and Toxicology 2020Quote: ... and a fourth group (DZP) received 2 mg/kg diazepam (CAS #439-14-5; Tocris, 2805; German-Ponciano et al., 2020) as a pharmacological control of anxiolytic activity ...
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bioRxiv - Physiology 2021Quote: ... Picrotoxin (100 µM) was used to block GABAA-receptor-mediated currents and D-2-amino-5-phosphonovalerate (APV; 20 µMm, Tocris Bioscience), and 6-cyano-7-nitroquinoxaline-2,3-dione (CNQX ...
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bioRxiv - Neuroscience 2022Quote: ... containing 10 μM 6-cyano-7-nitroquinoxaline-2,3-dione (CNQX) and 50 μM D,L-2-amino-5-phosphonovaleric acid (AP5) (both from Tocris, Bristol, UK) to block recurrent glutamatergic signaling.
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bioRxiv - Neuroscience 2023Quote: ... The following compounds were added to raCSF as indicated in the Results section: D-(-)-2-Amino-5-phosphonopentanoic acid (D-APV, 100 μM dissolved in H2O; Tocris Bioscience), (5S,10R)-(+)-5-Methyl-10,11-dihydro-5H-dibenzo[a,d] cyclohepten-5,10-imine maleate (MK-801 ...
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bioRxiv - Neuroscience 2024Quote: ... Both control and CACNA1A+/− networks at DIV49 were treated acutely with 100 µM D-2-amino-5-phosphonovalerate (D-AP5; Tocris, #0106) for 60 min ...
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bioRxiv - Molecular Biology 2020Quote: ... kin28as strains and their controls were then grown to an OD600 of 0.8 and treated with 6 μM of 1-Naphthyl PP1 (NAPP1; Tocris Bioscience) for 15 min ...
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bioRxiv - Neuroscience 2022Quote: Primary microglia cells from C57Bl/6 J mice cultured in presence of CSF-1 were treated with Formoterol (10 ng/ml, cat # 1448, Tocris) or vehicle for 1 hour ...
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bioRxiv - Cancer Biology 2023Quote: Around 1 x 105 cells were seeded in a 6-well plate for the drug treatment with Brequinar (Tocris, 6196) in a dose-dependent manner for 72 h ...
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bioRxiv - Biophysics 2021Quote: ... Cells were treated with 6 μM CHIR99021 (Tocris) for 48 hours on day 0 ...
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bioRxiv - Developmental Biology 2021Quote: ... 6 μM Chir 99021 (Tocris cat. no. 4423), 20ng/ml murine bFGF (PeproTech cat ...
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bioRxiv - Neuroscience 2020Quote: ... GABAA (6 µM bicuculline metiodide, Tocris, Bristol, UK) or GABAB (100 µM CGP46381 ...
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bioRxiv - Neuroscience 2020Quote: ... and Pyridone 6 (#6577) were purchased from Tocris Bioscience (Bristol ...
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bioRxiv - Neuroscience 2020Quote: ... 6-cyano-7-nitroquinoxaline-2,3-dione (CNQX, Tocris), 2,3-dihydroxy-6-nitro-7-sulfamoyl-benzo[f]quinoxaline-2,3-dione (NBQX ...
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bioRxiv - Molecular Biology 2020Quote: ... KN-62 and Inca-6 were from Tocris Bioscience (Minneapolis ...
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bioRxiv - Pharmacology and Toxicology 2021Quote: ... and SN-6 (2184) were purchased from Tocris, UK ...
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bioRxiv - Genetics 2021Quote: ... containing 6 μM or 12 μM CHIR99021 (Tocris) for 24 or 48 hours ...
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bioRxiv - Physiology 2023Quote: Xestospongin-C (Xe-C) -6 µM-(Tocris Bioscience). A membrane-permeably compound isolated from the sponge Xestospongia sp. ...
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bioRxiv - Genomics 2019Quote: ... On D3 medium was changed to 1:1 mix of spent and fresh RPMI Minus supplemented with 7.5μM IWP-2 (Tocris). On D5 ...
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bioRxiv - Neuroscience 2023Quote: ... Candidate ASM order information was as follows: 1-Ethyl-2-benzimidazolinone (Alternative name 1-EBIO, Tocris, CAS: 1041), AA43279 (Focus biomolecules ...
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bioRxiv - Neuroscience 2020Quote: ... mEPSCs were recorded for 5 min in the presence of 1 μM tetrodotoxin (Tocris), 10 μM CPP (Tocris) ...
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bioRxiv - Neuroscience 2023Quote: ... (-)-quinpirole HCl (QUIN; 0.05 mg/kg, 1 mg/kg or 5 mg/kg; Tocris), raclopride HCl (RACLO ...