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Citations for Tocris :
601 - 650 of 987 citations for 6 methyl 2 thioxo 2 3 dihydroquinazolin 4 1H one since 2019
Citations are collected from bioRxiv only, the total number of publications could be much larger.
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bioRxiv - Cell Biology 2022Quote: ... Inhibitors were resuspended in DMSO and serially diluted in medium to their final working concentration and added on day 0 (Lats1/2 inhibitor Truli40 (CSNpharm, # CSN26140) or the Limk1 inhibitor Damnacanthal41 (Tocris, # 1936)) ...
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bioRxiv - Neuroscience 2022Quote: ... Non-specific binding was measured in the presence of 2 µM of Xanthine Amine Congener (XAC, Tocris Bioscience, Bristol, United Kingdom), and the resulting values were subtracted from those obtained with [3H]DPCPX35 to determine the specific binding and normalized for protein concentration ...
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bioRxiv - Neuroscience 2023Quote: ... The following compounds were added to raCSF as indicated in the Results section: D-(-)-2-Amino-5-phosphonopentanoic acid (D-APV, 100 μM dissolved in H2O; Tocris Bioscience), (5S,10R)-(+)-5-Methyl-10,11-dihydro-5H-dibenzo[a,d] cyclohepten-5,10-imine maleate (MK-801 ...
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bioRxiv - Neuroscience 2023Quote: ... the medium was then changed to 3N (50:50 DMEM/F12:neurobasal with N2 and B27 supplements) without vitamin A with 2 µM DMH1 (Tocris, 4126), 2 µM XAV939 (Cayman Chemical ...
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bioRxiv - Physiology 2023Quote: ... the cell medium was replaced with the experimental medium (2 ml/well) consisting of DMEM containing 1 nM of 1,25-dihydroxyvitamin D3 (Tocris; Cat. #2551), as described previously58 ...
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bioRxiv - Neuroscience 2023Quote: iPSCs were replated at a density of 2 x 104 cells/cm2 in mTeSR medium containing 10 µM Rho kinase inhibitor (Y-27632, Tocris #5849), which was removed after 24 hours ...
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bioRxiv - Cell Biology 2024Quote: ... + 10 μM Tranylcypromine (2-PCPA) HCl (DMSO; Selleckchem S4246) + 20 μM Forskolin (DMSO; Selleckchem S2449) + 1 μM Ch 55 (DMSO; Tocris 2020) + 5 μM EPZ004777 (DMSO ...
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bioRxiv - Neuroscience 2024Quote: ... Both control and CACNA1A+/− networks at DIV49 were treated acutely with 100 µM D-2-amino-5-phosphonovalerate (D-AP5; Tocris, #0106) for 60 min ...
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bioRxiv - Cell Biology 2024Quote: ... 1.0×105 cells/cm2 for anti-fibrotic condition consisting in FibroGRO 2% FBS supplemented with 75ng/mL of bFGF and 500nM of TGF-β inhibitor (A83-01, Tocris). iPSC-cFbs were maintained for 7 days in culture replacing medium each second day ...
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bioRxiv - Immunology 2024Quote: ... The following inhibitors were added to the cells for 24 hours before harvesting: the NF-κB inhibitor JSH23 (2 µM, Tocris Bioscience), STING inhibitor H151 (5 µM ...
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bioRxiv - Cell Biology 2019Quote: ... 10µM 6-cyano-7-nitroquinoxaline-2,3-dione (CNQX; Tocris), and 50µM D-(-)-2-amino-5-phosphonopentanoic (D-AP5 or APV ...
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bioRxiv - Pharmacology and Toxicology 2023Quote: ... 8-Cyclopentyl-1,3-dipropylxanthine (DPCPX; Tocris, 102146-07-6), 4-[2-[[6-amino-9-(N-ethyl-β-D-ribofuranuronamidosyl)-9H-purin-2-yl]amino] ethyl]-benzenepropanoic acid ...
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bioRxiv - Neuroscience 2021Quote: ... The following chemical reagents were used: 4-aminopyridine (4-AP, TOCRIS, #940), ADX 71743 (TOCRIS ...
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bioRxiv - Neuroscience 2021Quote: ... 4-AP (Tocris, UK) was stored as a stock solution of 100 mM in ACSF at -20°C and applied to the bath at 5 mM ...
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bioRxiv - Developmental Biology 2021Quote: ... CHIR99021 (4 μM; Tocris), FGF2 (20 ng/mL ...
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bioRxiv - Cell Biology 2023Quote: ... 4-IPP (Tocris, 3429), and Brefeldin A (Millipore-Sigma ...
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bioRxiv - Genetics 2023Quote: ... 4 μM CHIR99021 (Tocris), 20 ng/mL FGF2 (PeproTech ...
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bioRxiv - Bioengineering 2021Quote: ... the medium was switched to N2B27 medium supplemented with 100 ng/mL VEGFA (ProSpec, CYT-116) and 2 μM forskolin (Tocris Bioscience, 1099) for two days ...
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bioRxiv - Neuroscience 2020Quote: ... containing 10 μM 6-cyano-7-nitroquinoxaline-2,3-dione (CNQX) and 50 μM D,L-2-amino-5-phosphonovaleric acid (AP5) to block glutamatergic signaling (both from Tocris, Bristol, UK). Experiments involving tetrodotoxin (TTX ...
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Transient upregulation of translational efficiency in prodromal Tg2576 mice precipitates AD symptomsbioRxiv - Neuroscience 2019Quote: Pharmacological inhibition of elF2α (eukaryotic translation initiation factor 2 subunit alpha) dephosphorylation was carried out by injecting salubrinal (Tocris Cat. No. 2347) emulsified in DMSO (Sigma ...
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bioRxiv - Cancer Biology 2024Quote: ... mice were randomized into groups and treated daily (5 days on, 2 days off) with 1mg/kg SB290157 trifluoroacetate (Tocris, 6860/5) intra-peritoneally ...
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bioRxiv - Neuroscience 2023Quote: ... in combination with potassium channel blocker 4-aminopyridine (4-AP, 1 mM, Tocris) to facilitate transmitter release at monosynaptic connections from RSC to ChC and recorded the PSP amplitudes (Figure 1H) ...
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bioRxiv - Neuroscience 2022Quote: ... 1 μM Pyr-3 (Tocris,3753), 1 mM MNI-caged-L-glutamate ...
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bioRxiv - Developmental Biology 2019Quote: ... and 3 μM CHIR99021 (Tocris Bioscience) for 3 days (after [13]) ...
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bioRxiv - Genomics 2021Quote: ... 3 μM CHIR99021 (Tocris, SML1046-5MG), 1000 U/mL ESGRO mLIF ...
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bioRxiv - Neuroscience 2022Quote: ... GABA (3 mM, Tocris Bioscience, 0344), CaCl2 (1.8 mM ...
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bioRxiv - Neuroscience 2023Quote: ... 3 mM CHIR-99021 (Tocris Biosciences), and 20 µM SB 431542 (Tocris Biosciences) ...
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bioRxiv - Molecular Biology 2023Quote: ... 3 μM CHIR 99021 (Tocris, 4423), and 50 nM PI 103 (Tocris ...
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bioRxiv - Molecular Biology 2023Quote: ... IPA-3 (Tocris, 3622, 5 μM), CK666 (Tocris ...
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bioRxiv - Developmental Biology 2023Quote: ... and 3 μM CHIR99021 (Tocris, 4423).
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bioRxiv - Neuroscience 2023Quote: ... and CHIR99021 3 μM (4423, Tocris). After 3 days ...
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bioRxiv - Developmental Biology 2023Quote: ... and 3 μM CHIR99021 (Tocris, 4423).
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bioRxiv - Molecular Biology 2023Quote: ... Ang II (4474-91-3, Tocris) was injected subcutaneously at a total dose of 1 ...
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bioRxiv - Neuroscience 2023Quote: ... 3 μM DCG-IV (Tocris Bioscience) was applied after each experiment ...
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bioRxiv - Bioengineering 2023Quote: ... and 3 µM CHIR99021 (Tocris Bioscience).
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bioRxiv - Molecular Biology 2024Quote: ... or NU-7441 (3 µM, Tocris) were added when specified 1 h prior to irradiation ...
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bioRxiv - Immunology 2022Quote: ... cells were treated with Pyridone 6 (Tocris Bioscience, Minneapolis, MN), Pimozide (Tocris Bioscience) ...
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bioRxiv - Neuroscience 2022Quote: ... 1 µM PKA inhibitor fragment (6-22) amide (Tocris Bioscience), 0.5 mM anisomycin (stock solution in EtOH ...
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bioRxiv - Neuroscience 2022Quote: ... 6-cyano-7-nitroquinoxaline-2,3-dione (CNQX, TOCRIS bioscience #0190), D,L-2-amino-5-phosphonovaleric acid (AP5 ...
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bioRxiv - Neuroscience 2020Quote: ... slices were equilibrated for 10 minutes while being continuously superfused at room temperature with oxygenated aCSF at 1-2 ml/min containing picrotoxin (50 μM, Tocris Bioscience, MO, USA) to block GABAA receptor-mediated inhibitory responses.
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bioRxiv - Neuroscience 2024Quote: ... a third group of animals were treated as those in group 2 with the addition of CB1 receptor antagonist AM251 (1 µM) (Tocris Bioscience, Bristol, UK). After 8 DIV ...
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bioRxiv - Neuroscience 2021Quote: ... 4-DAMP (Catalog #0482, Tocris), AFDX-384 (Catalog #1345 ...
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bioRxiv - Neuroscience 2019Quote: ... 4-AP (K channels; Tocris) JNJ-16259685 (mGluR1 ...
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bioRxiv - Immunology 2019Quote: ... 4-IPP (Tocris Catalog # 3429)43 ...
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bioRxiv - Cell Biology 2020Quote: ... KN-62 (4 μM, TOCRIS), BAPTA-AM (10 μM ...
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bioRxiv - Neuroscience 2021Quote: ... 4 µM SR 95531 (Tocris) and 10 µM DL-AP5 (Tocris) ...
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bioRxiv - Neuroscience 2023Quote: ... Topiramate (Tocris, #97240-79-4), and Carbamazepine (Tocris ...
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bioRxiv - Neuroscience 2023Quote: ... and 4 μM XAV (Tocris). On DIV 04 ...
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bioRxiv - Developmental Biology 2019Quote: ... 3 μM CHIR99021 (Tocris or Axon Medchem), 10 nM Retinoic Acid (Sigma) ...
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bioRxiv - Neuroscience 2020Quote: ... Dihydro-β-erythroidine (DhβE, 3 μM, Tocris) was used to block β2 containing nicotinic receptors ...