Glycerol Kinase 1 Blocking Peptidefrom Selleck Chemicals

TPI-1

TPI-1 (Tyrosine Phosphatase Inhibitor 1) is a potent inhibitor of SHP-1 with IC50 of 40 nM for...

Cat# S6570, SKU# S6570-25mg, 25mg, $497.00 Ask

HA14-1

HA14-1 is a non-peptidic ligand of a Bcl-2 surface pocket with IC50 of ~9 μM.

Cat# S1071, SKU# S1071-10mg, 10mg, $79.00 Ask

NQDI-1

NQDI 1, an inhibitor of ASK1(apoptosis signal-regulating kinase 1), attenuates acute ischemic...

Cat# S8289, SKU# S8289-10mg, 10mg, $97.00 Ask

1-Hexadecanol

1-Hexadecanol is a fatty alcohol used to make other chemicals.

Cat# S4173, SKU# S4173-50mg, 50mg, $97.00 Ask

1-Furfurylpyrrole

1-Furfurylpyrrole (N-Furfurylpyrrole) is a potential contributor of flavor and aroma to popcorn.

Cat# S6107, SKU# S6107-25ul, 25ul, $97.00 Ask

HOIPIN-1

HOIPIN-1 (JTP-0819958, HOIP inhibitor-1) is a linear ubiquitin chain assembly complex (LUBAC)...

Cat# S6396, SKU# S6396-25mg, 25mg, $657.00 Ask

PAC-1

PAC-1 is a potent procaspase-3 activator with EC50 of 0.22 μM and the first small molecule known...

Cat# S2738, SKU# S2738-10mM/1mL, 10mM/1mL, $120.00 Ask

BTB-1

BTB-1 is a novel, selective and reversible inhibitor of the mitotic motor protein Kif18A with...

Cat# S6796, SKU# S6796-25mg, 25mg, $177.00 Ask

A2ti-1

A2ti-1 is a selective and high-affinity inhibitor of annexin A2/S100A10 heterotetramer (A2t)...

Cat# E1421, SKU# E1421-25mg, 25mg, $890.00 Ask

BH3I-1

BH3I-1 is a Bcl-XL-BH3 domain interaction inhibitor with Ki of 2.4 μM (by fluorescence...

Cat# S8177, SKU# S8177-5mg, 5mg, $97.00 Ask

Leukadherin-1

Leukadherin-1 (LA1) is a small molecule agonist that enhances CD11b/CD18-dependent cell adhesion...

Cat# S8306, SKU# S8306-10mg, 10mg, $97.00 Ask

TRi-1

TRi-1 (HUN20688, TXNRD1 inhibitor 1) is a potent, specific and irreversible cytosolic...

Cat# S0267, SKU# S0267-5mg, 5mg, $187.00 Ask

NGI-1

NGI-1 is an aminobenzamide-sulfonamide compound that targets both oligosaccharyltransferase...

Cat# S8750, SKU# S8750-10mg, 10mg, $97.00 Ask

TAI-1

TAI-1 is a potent and specific Hec1 inhibitor, which disrupts Hec1-Nek2 protein interaction.

Cat# S7495, SKU# S7495-25mg, 25mg, $477.00 Ask

Mdivi-1

Mdivi-1 (Mitochondrial division inhibitor 1) is a selective cell-permeable inhibitor of...

Cat# S7162, SKU# S7162-20mg, 20mg, $147.00 Ask

BTZO-1

BTZO-1 binds to macrophage migration inhibitory factor (MIF) with Kd of 68.6 nM. BTZO-1 activats...

Cat# S0539, SKU# S0539-25mg, 25mg, $417.00 Ask

Alda 1

Alda 1 is an ALDH2 agonist that activates catalysis for both wild-type ALDH2 (ALDH2*1) and ALDH2*2.

Cat# S5800, SKU# S5800-25mg, 25mg, $290.00 Ask

TAPI-1

TAPI-1 is an ADAM17/TACE inhibitor, which blocks shedding of cytokine receptors. TAPI-1 is also...

Cat# S7434, SKU# S7434-10mM/1mL, 10mM/1mL, $1190.00 Ask

Cited in: Targeting neuronal activity-regulated neuroligin-3 dependency for high-grade glioma therapy

Humsa S. Venkatesh, et al., bioRxiv - Neuroscience 2017

Quote: ... TAPI-1 at 20uM (ADAM17 inhibitor; S7434; Selleck Chemicals); GI 254023X at 200nM (ADAM10 inhibitor ...

Oncrasin-1

Oncrasin-1 (Onc-1) is a potent RNA polymerase II inhibitor with antitumor activity that kills...

Cat# S0780, SKU# S0780-25mg, 25mg, $297.00 Ask

BLT-1

BLT-1(Block lipid transport-1), a thiosemicarbazone copper chelator, is a selective inhibitor of...

Cat# S0857, SKU# S0857-25mg, 25mg, $687.00 Ask

Shield-1

Shield-1 is a specific, cell-permeant and high-affinity ligand of FK506-binding protein-12...

Cat# S3469, SKU# S3469-25mg, 25mg, $1470.00 Ask

G-1

G-1 (LNS 8801) is a nonsteroidal and selective agonist of G protein-coupled receptor 30 (GPR30,...

Cat# S0851, SKU# S0851-10mM/1mL, 10mM/1mL, $439.00 Ask

IMR-1

IMR-1 is a novel class of Notch inhibitors targeting the transcriptional activation with IC50 of 26 μM.

Cat# S8280, SKU# S8280-5mg, 5mg, $117.00 Ask

Spautin-1

Spautin-1 is a potent and specific autophagy inhibitor, and inhibits the deubiquitinating...

Cat# S7888, SKU# S7888-50mg, 50mg, $447.00 Ask

JANEX-1

JANEX-1 (WHI-P131) is a small molecule inhibitor of JAK3 that selectively inhibits JAK3 at an...

Cat# S5903, SKU# S5903-25mg, 25mg, $397.00 Ask

TPI-1

TPI-1 (Tyrosine Phosphatase Inhibitor 1) is a potent inhibitor of SHP-1 with IC50 of 40 nM for...

Cat# S6570, SKU# S6570-10mM/1mL, 10mM/1mL, $177.00 Ask

1-Octacosanol

1-Octacosanol (n-Octacosanol, Octacosyl alcohol, Octanosol, Montanyl alcohol, Cluytyl alcohol)...

Cat# S5161, SKU# S5161-25mg, 25mg, $97.00 Ask

4EGI-1

4EGI-1 is a competitive eIF4E/eIF4G interaction inhibitor by binding to eIF4E with KD of 25 μM....

Cat# S7369, SKU# S7369-100mg, 100mg, $777.00 Ask

Cited in: Ribosome Quality Control Mechanism Mitigates the Cytotoxic Impacts of Ribosome Collisions Induced by 5-Fluorouracil

Susanta Chatterjee, et al., bioRxiv - Cell Biology 2023

Quote: ... or 25 μM 4EGI-1 (Selleck Chemicals, Cat. # S7369) for 24 h before incubation with 2.5 μM of 5FU for the indicated time-points ...

G6PDi-1

G6PDi-1 is an effective inhibitor of glucose-6-phosphate dehydrogenase (G6PD). G6PDi-1 depletes...

Cat# S9617, SKU# S9617-5mg, 5mg, $270.00 Ask

1-Phenylbiguanide

1-Phenylbiguanide (Phenylbiguanide, PBG, N-Phenylbiguanide) is a 5-hydroxytryptamine3 (5-HT3)...

Cat# S2578, SKU# S2578-25mg, 25mg, $97.00 Ask

Necrostatin-1

Necrostatin-1 (Nec-1) is a specific RIP1 (RIPK1) inhibitor and inhibits TNF-α-induced...

Cat# S8037, SKU# S8037-1g, 1g, $970.00 Ask

Cited in: Acid Ceramidase Inhibitor LCL-805 Antagonizes Akt Signaling and Promotes Iron-Dependent Cell Death in Acute Myeloid Leukemia

Johnson Ung, et al., bioRxiv - Cancer Biology 2023

Quote: ... necrostatin-1 (Selleck Chemicals, #S8037); pepstatin A (Cayman ...

TPCA-1

TPCA-1 (GW683965) is an inhibitor of IKK-2 with IC50 of 17.9 nM in a cell-free assay, inhibits...

Cat# S2824, SKU# S2824-10mM/1mL, 10mM/1mL, $220.00 Ask

HOIPIN-1

HOIPIN-1 (JTP-0819958, HOIP inhibitor-1) is a linear ubiquitin chain assembly complex (LUBAC)...

Cat# S6396, SKU# S6396-5mg, 5mg, $217.00 Ask

Apostatin-1

Apostatin-1 (Apt-1) is a novel TRADD inhibitor. Apostatin-1 binds to a pocket on the N-terminal...

Cat# S9705, SKU# S9705-5mg, 5mg, $157.00 Ask

PAC-1

PAC-1 is a potent procaspase-3 activator with EC50 of 0.22 μM and the first small molecule known...

Cat# S2738, SKU# S2738-10mg, 10mg, $90.00 Ask

MZ-1

MZ-1 is a PROTAC degrader of bromodomain-containing protein 4 (BRD4). MZ-1 binds to the Brd...

Cat# S8889, SKU# S8889-5mg, 5mg, $217.00 Ask

JC-1

JC-1 (CBIC2, NK 1420), a fluorescent lipophilic carbocyanine dye, is a mitochondrial potential...

Cat# S9784, SKU# S9784-5mg, 5mg, $427.00 Ask

Torin 1

Torin 1 is a potent inhibitor of mTORC1/2 with IC50 of 2 nM/10 nM in cell-free assays; exhibits...

Cat# S2827, SKU# S2827-200mg, 200mg, $1870.00 Ask

Cited in: Adaptation of pancreatic cancer cells to nutrient deprivation is reversible and requires glutamine synthetase stabilization by mTORC1

Pei-Yun Tsai, et al., bioRxiv - Cancer Biology 2020

Quote: ... Torin 1 (Selleck Chemicals, S2827).

» View all citations

Vacuolin-1

Vacuolin-1 is a potent and cell-permeable inhibitor that blocks the Ca(2+)-dependent exocytosis...

Cat# S6912, SKU# S6912-10mM/1mL, 10mM/1mL, $137.00 Ask

BMS-1

BMS-1 is a small-molecule inhibitor of PD-1/PD-L1 interaction with IC50 of 6 nM.

Cat# S7911, SKU# S7911-25mg, 25mg, $497.00 Ask

TPCA-1

TPCA-1 (GW683965) is an inhibitor of IKK-2 with IC50 of 17.9 nM in a cell-free assay, inhibits...

Cat# S2824, SKU# S2824-10mg, 10mg, $170.00 Ask

FSL-1

FSL-1, a bacterial-derived toll-like receptor 2/6 (TLR2/6) agonist, enhances resistance to...

Cat# S8428, SKU# S8428-5mg, 5mg, $927.00 Ask

ITD-1

ITD-1 is a potent TGF-β inhibitor. It does not block the kinase activity of either type I...

Cat# S6713, SKU# S6713-10mM/1mL, 10mM/1mL, $117.00 Ask

HA14-1

HA14-1 is a non-peptidic ligand of a Bcl-2 surface pocket with IC50 of ~9 μM.

Cat# S1071, SKU# S1071-50mg, 50mg, $170.00 Ask

Liproxstatin-1

Liproxstatin-1 is a potent ferroptosis inhibitor with an IC50 of 22 nM.

Cat# S7699, SKU# S7699-100mg, 100mg, $997.00 Ask

Cited in: Acid Ceramidase Inhibitor LCL-805 Antagonizes Akt Signaling and Promotes Iron-Dependent Cell Death in Acute Myeloid Leukemia

Johnson Ung, et al., bioRxiv - Cancer Biology 2023

Quote: ... liproxstatin-1 (Selleck Chemicals, #S7699); ferrostatin-1 (Selleck Chemicals ...

TAPI-1

TAPI-1 is an ADAM17/TACE inhibitor, which blocks shedding of cytokine receptors. TAPI-1 is also...

Cat# S7434, SKU# S7434-1mg, 1mg, $270.00 Ask

Cited in: Targeting neuronal activity-regulated neuroligin-3 dependency for high-grade glioma therapy

Humsa S. Venkatesh, et al., bioRxiv - Neuroscience 2017

Quote: ... TAPI-1 at 20uM (ADAM17 inhibitor; S7434; Selleck Chemicals); GI 254023X at 200nM (ADAM10 inhibitor ...

Torin 1

Torin 1 is a potent inhibitor of mTORC1/2 with IC50 of 2 nM/10 nM in cell-free assays; exhibits...

Cat# S2827, SKU# S2827-10mg, 10mg, $170.00 Ask

Cited in: Adaptation of pancreatic cancer cells to nutrient deprivation is reversible and requires glutamine synthetase stabilization by mTORC1

Pei-Yun Tsai, et al., bioRxiv - Cancer Biology 2020

Quote: ... Torin 1 (Selleck Chemicals, S2827).

» View all citations

WQ 1

WQ 1 is a high affinity and selective σ1 receptor antagonist with pKi values of 10.85, 6.53 and...

Cat# E0388, SKU# E0388-5mg, 5mg, $227.00 Ask

AMI-1

AMI-1 is a potent and specific Histone Methyltransferase (HMT) inhibitor with IC50 of 3.0 μM and...

Cat# S7884, SKU# S7884-10mM/1mL, 10mM/1mL, $117.00 Ask

RCM-1

RCM-1 is a nontoxic inhibitor of Forkhead box M1 (FOXM1) that suppresses goblet cell metaplasia...

Cat# S6898, SKU# S6898-25mg, 25mg, $717.00 Ask

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