Sigma-1 receptor antagonist 3

Supplier MedChemExpress
Product # HY-125820-50 mg
CAS # 1639220-17-9
Pricing 50 mg, USD $1450.0
Biological Activity Sigma-1 receptor antagonist 3 (compound135) is a potent and selective Sigma-1 (σ1) receptor antagonist with a Ki of 1.14 nM. Sigma-1 receptor antagonist 3 inhibits Human Ether-a-go-go-Related Gene (hERG) with an IC50 of 1.54 μM. Sigma-1 receptor antagonist 3 has the potential for the neuropathic pain[1].
Purity 99.47%
MWt 363.86
Formula C₁₉H₂₃ClFN₃O
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