Sigma-1 receptor antagonist 3
Supplier | MedChemExpress |
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Product # | HY-125820-50 mg |
CAS # | 1639220-17-9 |
Pricing | 50 mg, USD $1450.0 |
Biological Activity | Sigma-1 receptor antagonist 3 (compound135) is a potent and selective Sigma-1 (σ1) receptor antagonist with a Ki of 1.14 nM. Sigma-1 receptor antagonist 3 inhibits Human Ether-a-go-go-Related Gene (hERG) with an IC50 of 1.54 μM. Sigma-1 receptor antagonist 3 has the potential for the neuropathic pain[1]. |
Purity | 99.47% |
MWt | 363.86 |
Formula | C₁₉H₂₃ClFN₃O |