PKA Inhibitor Fragment (6-22) amide
Supplier | MedChemExpress |
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Product # | HY-P1290 |
CAS # | 121932-06-7 |
Pricing | inquire |
Biological Activity | PKA Inhibitor Fragment (6-22) amide is an inhibitor of cAMP-dependent protein kinase A (PKA), with a Ki of 2.8 nM. PKA Inhibitor Fragment (6-22) amide can significantly reverse low-level morphine antinociceptive tolerance in mice[1][2]. |
Synonyms | PKI-(6-22)-amide |
MWt | 1868.06 |
Formula | C₈₀H₁₃₀N₂₈O₂₄ |