Lck Inhibitor
Lck Inhibitor is a small-molecule inhibitor. It takes participate in the T-cell receptor (TCR) signal transduction and affects the expression of genes associated with cell proliferation, cytokine release and T-cell survival. It has been designed and developed as therapeutic agents for the treatment for T-cell-mediated autoimmune and organ transplant rejection. It showed high selectivity against Lck over another Src family kinase Src and the kinases. It also showed more than 1000-fold greater selectivity over CDK, MAPK and the RSK family.
| Supplier | BOC Sciences |
|---|---|
| Product # | 847950-09-8 |
| Pricing | Inquire |
| Cas | 847950-09-8 |
| Molecular Weight | 530.62 |
| Molecular Formula | C31H30N8O |
| Canonical SMILES | CC1=C(C(=CC=C1)C)N2C(=O)C3=CN=C(N=C3N4C2=NC5=CC=CC=C54)NC6=CC=C(C=C6)N7CCN(CC7)C |