AR-A 2
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-107018 |
| CAS # | 220051-79-6 |
| Pricing | inquire |
| Biological Activity | AR-A 2 is a selective 5-HT1B receptor antagonist, with high affinity to guinea pig cortex 5HT1B/1D and recombinant guinea pig 5-HT1B receptors (Ki=0.24 and 0.47 nM) and with 10-fold lower affinity to guinea pig 5-HT1D receptor (Ki, 5 nM), and shows an EC50 of 4.5 nM for the guinea pig 5-HT1B receptor; AR-A 2 can be used in the research of depression and anxiety. |
| Synonyms | AR-A 000002 |
| MWt | 448.6 |
| Formula | C₂₇H₃₆N₄O₂ |