GCN2-IN-6
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-130240-100 mg |
| CAS # | 2183470-09-7 |
| Pricing | 100 mg, USD $2800.0 |
| Biological Activity | GCN2-IN-6 (Compound 6d) is a potent, and orally available GCN2 inhibitor confirmed by in-house enzymatic (IC50 of 1.8 nM) and cellular assays (IC50 of 9.3 nM). GCN2-IN-6 is also a eIF2α kinase PERK inhibitor with an IC50 of 0.26 nM (in enzymatic assay) and 230 nM (in cells)[1]. |
| Purity | 98.47% |
| MWt | 485.29 |
| Formula | C₁₉H₁₂Cl₂F₂N₄O₃S |