Apelin-36(human) TFA
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-P1064A |
| Pricing | inquire |
| Biological Activity | Apelin-36(human) TFA is an endogenous orphan G protein-coupled receptor APJ agonist, with an EC50 of 20 nM. Apelin-36(human) TFA shows high affinity to human APJ receptors expressed in HEK 293 cells (pIC550=8.61). Apelin-36(human) TFA has been linked to two major types of biological activities: cardiovascular and metabolic. Apelin-36(human) TFA inhibits the entry of some HIV-1 and HIV-2 into the NP2/CD4 cells expressing APJ[1][2][3][4]. |
| MWt | 4309.85 |
| Formula | C₁₈₆H₂₉₈F₃N₆₉O₄₅S |