SB 243213 dihydrochloride
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-103112A |
| CAS # | 1780372-25-9 |
| Pricing | inquire |
| Biological Activity | SB 243213 dihydrochloride is an orally active, selective and high-affinity 5-HT2C receptor antagonist with a pKi of 9.37 and a pKb of 9.8 for human 5-HT2C receptor. SB 243213 dihydrochloride shows greater than a 100-fold selectivity over a wide range of neurotransmitter receptors, enzymes and ion channels. SB 243213 dihydrochloride has improved anxiolytic profile and has the potential for schizophrenia and motor disorders[1]. |
| Purity | ≥99.0% |
| MWt | 501.33 |
| Formula | C₂₂H₂₁Cl₂F₃N₄O₂ |