(E/Z)-GSK5182

Supplier MedChemExpress
Product # HY-111226A-100 mg
Pricing 100 mg, USD $1800.0
Biological Activity (E/Z)-GSK5182 is a racemic compound of (E)-GSK5182 and (Z)-GSK5182 isomers. GSK5182 is a highly selective and orally active inverse agonist of estrogen-related receptor γ (ERRγ) with an IC50 of 79 nM[1]. GSK5182 also induces reactive oxyen species (ROS) generation in hepatocellular carcinoma[1][2][3].
Purity 98.90%
MWt 417.54
Formula C₂₇H₃₁NO₃
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