Alvimopan monohydrate

Supplier MedChemExpress
Product # HY-76657-2 mg
CAS # 1383577-62-5
Pricing 2 mg, USD $80.0
Synonyms ADL 8-2698 monohydrate; LY 246736 monohydrate
MWt 442.55
Formula C₂₅H₃₄N₂O₅
Biological Activity Alvimopan monohydrate (ADL 8-2698 monohydrate) is a potent, selective, orally active and reversible μ-opioid receptor antagonist, with an IC50 of 1.7 nM. Alvimopan monohydrate has selectivity for μ-opioid receptor (Ki=0.47 nM) over κ- and δ-opioid receptors (Kis=100, 12 nM, respectively). Alvimopan monohydrate can be used for the research of postoperative ileus[1][2][3].
Purity 99.18%
Feedback