Alvimopan monohydrate
Supplier | MedChemExpress |
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Product # | HY-76657-2 mg |
CAS # | 1383577-62-5 |
Pricing | 2 mg, USD $80.0 |
Synonyms | ADL 8-2698 monohydrate; LY 246736 monohydrate |
MWt | 442.55 |
Formula | C₂₅H₃₄N₂O₅ |
Biological Activity | Alvimopan monohydrate (ADL 8-2698 monohydrate) is a potent, selective, orally active and reversible μ-opioid receptor antagonist, with an IC50 of 1.7 nM. Alvimopan monohydrate has selectivity for μ-opioid receptor (Ki=0.47 nM) over κ- and δ-opioid receptors (Kis=100, 12 nM, respectively). Alvimopan monohydrate can be used for the research of postoperative ileus[1][2][3]. |
Purity | 99.18% |