GN 44028
GN 44028 is a potent HIF-1α inhibitor (IC50 = 14 nM). It suppresses hypoxia-induced HIF-1α transcriptional activity with no effect on HIF-1α mRNA expression, HIF-1α protein accumulation, or HIF-1α/HIF-1β heterodimerization.
Supplier | BOC Sciences |
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Product # | 1421448-26-1 |
Pricing | Inquire |
Cas | 1421448-26-1 |
Molecular Weight | 305.33 |
Molecular Formula | C18N15N3O2 |
Canonical SMILES | C1COC2=C(O1)C=CC(=C2)NC3=NNC4=C3CC5=CC=CC=C54 |