RG108

Supplier MedChemExpress
Product # HY-13642-10 mg
CAS # 48208-26-0
Pricing 10 mg, USD $72.0
Synonyms N-Phthalyl-L-tryptophan
MWt 334.33
Formula C₁₉H₁₄N₂O₄
Biological Activity RG108 (N-Phthalyl-L-tryptophan) is a non-nucleoside DNA methyltransferases (DNMTs) inhibitor (IC50=115 nM) that blocks the DNMTs active site. RG108 (N-Phthalyl-L-tryptophan) causes demethylation and reactivation of tumor suppressor genes, but it does not affect the methylation of centromeric satellite sequences[1][2][3].
Purity 99.81%
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