GYKI 52466 dihydrochloride
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-103234A-10 mg |
| CAS # | 2319722-40-0 |
| Pricing | 10 mg, inquire |
| Biological Activity | GYKI 52466 dihydrochloride is a potent, selective, orally active and non-competitive kainate- and AMPA-activated currents antagonist with IC50s of 7.5 μM and 11 μM, respectively. GYKI 52466 dihydrochloride is inactive against N-methyl-D-aspartate (NMDA) or γ-aminobutyric acid responses. GYKI 52466 dihydrochloride ia a muscle relaxant and anticonvulsant agent, and has good blood brain barrier permeability[1][2]. |
| MWt | 366.24 |
| Formula | C₁₇H₁₇Cl₂N₃O₂ |