A-582941 dihydrochloride
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-59201A |
| CAS # | 848591-90-2 |
| Pricing | inquire |
| Biological Activity | A-582941 dihydrochloride is a potent, selective and brain-penetrant partial agonist of α7 nAChR, with Kis of 10.8 and 16.7 nM in rat brain membranes and human frontal cortex, respectively. A-582941 dihydrochloride also binds to human 5-HT3 receptor with a Ki of 150 nM. A-582941 has the potential for cognitive deficits associated with various neurodegenerative and psychiatric disorders research[1][2]. |
| MWt | 353.29 |
| Formula | C₁₇H₂₂Cl₂N₄ |