Vernakalant Hydrochloride

Supplier MedChemExpress
Product # HY-14183-2 mg
CAS # 748810-28-8
Pricing 2 mg, USD $180.0
Biological Activity Vernakalant hydrochloride is a mixed voltage- and frequency-dependent Na+ and atria-preferred K+ channel blocker. IC50 for block by Vernakalant of wild-type and mutant Kv1.5 channels Fractional block is 13.35±0.93 μM, 0.61±0.03 μM, and 1.63±0.09 μM for Kv1.5 channelwt, Kv1.5 channelI508F, Kv1.5 channelT479A, respectively.
Synonyms RSD1235 hydrochloride
MWt 385.93
Formula C₂₀H₃₂ClNO₄
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