GATA4-NKX2-5-IN-1
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-103484 |
| CAS # | 544681-96-1 |
| Pricing | inquire |
| Biological Activity | GATA4-NKX2-5-IN-1 (Compound 3) dose-dependently inhibits the GATA4–NKX2-5 transcriptional synergy with an IC50 of 3 μM. GATA4-NKX2-5-IN-1 exhibits no activity on the protein kinases involved in the regulation of GATA4 phosphorylation, and it modulates the hypertrophic agonist-induced cardiac gene expression[1]. |
| MWt | 349.43 |
| Formula | C₂₁H₂₃N₃O₂ |