Gaboxadol hydrochloride

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Supplier MedChemExpress
Product # HY-10233-50 mg
CAS # 85118-33-8
Pricing 50 mg, USD $120.0
Synonyms Lu 02-030 hydrochloride; THIP hydrochloride
MWt 176.6
Formula C₆H₉ClN₂O₂
Biological Activity
  • Gaboxadol hydrochloride (Lu 02-030 hydrochloride; THIP hydrochloride) is a potent agonist of the GABAA receptor and an antagonist of GABAC receptors (IC50=25 μM). Gaboxadol hydrochloride displays
  • a partial agonist efficacy on subunit α1β2γ2 with an ED50 value of 143 µM, a full agonist efficacy at α5 subunit (ED50=28-129 µM) and a superagonist efficacy at α4β3δ (ED50=6 µM). Gaboxadol hydrochloride is a non-opioid analgesic and has hypnotic activities[1][2].
Purity ≥98.0%
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