WAY-181187
Supplier | MedChemExpress |
---|---|
Product # | HY-14340-10 mg |
CAS # | 554403-49-5 |
Pricing | 10 mg, USD $550.0 |
Synonyms | SAX-187 |
MWt | 380.87 |
Formula | C₁₅H₁₃ClN₄O₂S₂ |
Biological Activity | WAY-181187 (SAX-187) is a potent and selective full 5-HT6 receptor agonist with a Ki of 2.2 nM and an EC50 of 6.6 nM[1]. WAY181187 mediates 5-HT6 receptor-dependent signal pathways, such as cAMP, Fyn and ERK1/2 kinase, as specific agonist[2]. |
Purity | 98.05% |