6-Iodonordihydrocapsaicin
6-Iodonordihydrocapsaicin is a potent and competitive vanilloid TRPV1 (VR1) receptor antagonist with IC50 value of 10 nM. It inhibits capsaicin-induced [Ca2+]i increase in rat DRG neurons. It also inhibits guinea pig bladder and trachea contractions in vitro. It may induce luciferase gene expression.
Supplier | BOC Sciences |
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Product # | 859171-97-4 |
Pricing | Inquire |
Cas | 859171-97-4 |
Molecular Weight | 419.30 |
Molecular Formula | C17H26INO3 |
Canonical SMILES | CCCCCCCCC(=O)NCC1=CC(=C(C=C1I)O)OC |