PKCβ inhibitor 1
Supplier | MedChemExpress |
---|---|
Product # | HY-13335-1 mg |
CAS # | 257879-35-9 |
Pricing | 1 mg, USD $275.0 |
Biological Activity | PKCβ inhibitor 1 is a potent, ATP-competitive, and selective PKCβ inhibitor with IC50s of 21 and 5 nM for human PKCβ1 and PKCβ2, respectively. PKCβ inhibitor 1 exhibits selectivity of more than 60-fold in favor of PKCβ2 relative to other PKC isozymes (PKCα, PKCγ, and PKCε)[1][2]. |
Purity | 98.21% |
MWt | 411.46 |
Formula | C₂₄H₂₁N₅O₂ |