Keap1-Nrf2-IN-1

Supplier MedChemExpress
Product # HY-126245-5 mg
CAS # 2232112-72-8
Pricing 5 mg, USD $450.0
Biological Activity Keap1-Nrf2-IN-1 is a Keap1 (Kelch-like ECH-associated protein 1)-Nrf2 (nuclear factor erythroid 2-related factor 2) protein-protein interaction inhibitor, and with an IC50 of 43 nM for Keap1 protein. Keap1-Nrf2-IN-1 activates Nrf2-regulated cytoprotective response and antagonizes Acetaminophen-induced liver injury[1].
Purity 98.08%
MWt 484.52
Formula C₂₄H₂₄N₂O₇S
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