GSK484 hydrochloride

Supplier MedChemExpress
Product # HY-100514-25 mg
CAS # 1652591-81-5
Pricing 25 mg, USD $590.0
Biological Activity GSK484 hydrochloride is a selective and reversible peptidylarginine deiminase 4 (PAD4) inhibitor. GSK484 hydrochloride demonstrates high affinity binding to PAD4 with IC50s of 50 nM in the absence of Calcium. In the presence of 2 mM Calcium, notably lower potency (250 nM) is observed.
MWt 510.03
Formula C₂₇H₃₂ClN₅O₃
Feedback