GSK484 hydrochloride
Supplier | MedChemExpress |
---|---|
Product # | HY-100514-25 mg |
CAS # | 1652591-81-5 |
Pricing | 25 mg, USD $590.0 |
Biological Activity | GSK484 hydrochloride is a selective and reversible peptidylarginine deiminase 4 (PAD4) inhibitor. GSK484 hydrochloride demonstrates high affinity binding to PAD4 with IC50s of 50 nM in the absence of Calcium. In the presence of 2 mM Calcium, notably lower potency (250 nM) is observed. |
MWt | 510.03 |
Formula | C₂₇H₃₂ClN₅O₃ |