Asimadoline hydrochloride
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-107384A-5 mg |
| CAS # | 185951-07-9 |
| Pricing | 5 mg, USD $84.0 |
| Synonyms | EMD-61753 hydrochloride |
| MWt | 451.0 |
| Formula | C₂₇H₃₁ClN₂O₂ |
| Biological Activity | Asimadoline (EMD-61753) hydrochloride is an orally active, selective and peripherally active κ-opioid agonist with IC50s of 5.6 nM (guinea pig) and 1.2 nM (human recombinant). Asimadoline hydrochloride has low permeability across the blood brain barrier and has peripheral anti-inflammatory actions. Asimadoline hydrochloride ameliorates allodynia in diabetic rats and has the potential for irritable bowel syndrome (IBS)[1][2][3]. |
| Purity | 99.80% |