Pizotifen malate
Pizotifen, also known as Pizotyline, is a benzocycloheptene-based drug used as a medicine, primarily as a preventative to reduce the frequency of recurrent migraine headaches. Pizotifen is a serotonin antagonist acting mainly at the 5-HT2A and 5HT2C receptors. It also has some activity as an antihistamine as well as some anticholinergic activity.
| Supplier | Ace Therapeutics |
|---|---|
| Product # | SMD1109 |
| CAS # | 5189-11-7 (malate) |
| Pricing | Customizable size, Inquiry |
| Synonym | Pizotyline malate; BC-105 malate; Litec malate; Pizotifen malate; Sanomtgran. |
| Product Category | Lab-use Small Molecule Drugs |
| Chemical Formula | C23H27NO5S |
| Molecular Weight | 429.531 |
| Elemental Analysis | C, 64.32; H, 6.34; N, 3.26; O, 18.62; S, 7.46 |
| IUPAC/Chemical Name | 4-(9,10-dihydro-4H-benzo[4,5]cyclohepta[1,2-b]thiophen-4-ylidene)-1-methylpiperidine malate |
| InChi Key | IWAWCPZVTXCFKD-UHFFFAOYSA-N |
| InChi Code | InChI=1S/C19H21NS.C4H6O5/c1-20-11-8-15(9-12-20)19-16-5-3-2-4-14(16)6-7-18-17(19)10-13-21-18;5-2(4(8)9)1-3(6)7/h2-5,10,13H,6-9,11-12H2,1H3;2,5H,1H2,(H,6,7)(H,8,9) |
| SMILES Code | CN1CC/C(CC1)=C2C3=CC=CC=C3CCC4=C\2C=CS4.OC(CC(O)=O)C(O)=O |
| Appearance | Solid powder |
| Purity | >98% (or refer to the Certificate of Analysis) |
| Shipping Condition | Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs. |
| Storage Condition | Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years). |
| Solubility | Soluble in DMSO |
| Shelf Life | >2 years if stored properly |
| Drug Formulation | This drug may be formulated in DMSO |
| Stock Solution Storage | 0 - 4℃ for short term (days to weeks), or -20℃ for long term (months). |
| HS Tariff Code | 2934.99.9001 |
| Availability | 2 Weeks |