(Rac)-Tavapadon
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-119486A-10 mM * 1 mL |
| CAS # | 1643462-64-9 |
| Pricing | 10 mM * 1 mL, USD $165.0 |
| Synonyms | (Rac)-PF-06649751; (Rac)-CVL-751 |
| MWt | 391.34 |
| Formula | C₁₉H₁₆F₃N₃O₃ |
| Biological Activity | (Rac)-Tavapadon ((Rac)-PF-06649751) is a potent and selective noncatechol dopamine D1 receptor agonist. (Rac)-Tavapadon displays potent full agonism in the GS activation assay as well as partial agonism in the β-arrestin2 recruitment assay (GS-cAMP, EC50=0.8 nM; β-arrestin2, EC50=68 nM). (Rac)-Tavapadon has antiparkinsonian activity[1]. |
| Purity | 99.63% |