Jaspamycin
Supplier | MedChemExpress |
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Product # | HY-111759-100 mg |
CAS # | 22242-96-2 |
Pricing | 100 mg, USD $2250.0 |
Synonyms | 7-CN-7-C-Ino |
MWt | 292.25 |
Formula | C₁₂H₁₂N₄O₅ |
Biological Activity | Jaspamycin (7-CN-7-C-Ino) is a potent activator of PKA, binding to the R site (PKAR), with an EC50 of 6.5 nM and Kd of 8 nM in Trypanosoma brucei. Jaspamycin (7-CN-7-C-Ino) does not bind with purified human PKARIα. Anti-parasite activity[1]. |
Purity | 98.73% |