(R)-PS210
Supplier | MedChemExpress |
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Product # | HY-13856 |
CAS # | 1410101-89-1 |
Pricing | inquire |
Biological Activity | (R)-PS210, the R enantiomer of PS210 (compound 4h-eutomer), is a substrate-selective allosteric activator of PDK1 with an AC50 value of 1.8 μM. (R)-PS210 targets to the PIF-binding pocket of PDK1. PIF: The protein kinase C-related kinase 2 (PRK2)-interacting fragment[1]. |
MWt | 380.31 |
Formula | C₁₉H₁₅F₃O₅ |