L-732138

Supplier MedChemExpress
Product # HY-101249-1 mg
CAS # 148451-96-1
Pricing 1 mg, USD $85.0
Biological Activity L-732138 is a selective, potent and competitive neurokinin-1 (NK-1) receptor antagonist with an IC50 of 2.3 nM. L-732138 has 200-fold more potent in cloned human NK-1 receptors than cloned rat NK-1 receptors, and has > 1000-fold more potent than human NK-2 and NK-3 receptors. L-732138 can reduce hyperalgesia and has antitumor action[1][2].
Purity ≥99.0%
MWt 472.38
Formula C₂₂H₁₈F₆N₂O₃
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