(E/Z)-GSK5182
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-111226A-10 mM * 1 mL |
| Pricing | 10 mM * 1 mL, USD $308.0 |
| Biological Activity | (E/Z)-GSK5182 is a racemic compound of (E)-GSK5182 and (Z)-GSK5182 isomers. GSK5182 is a highly selective and orally active inverse agonist of estrogen-related receptor γ (ERRγ) with an IC50 of 79 nM[1]. GSK5182 also induces reactive oxyen species (ROS) generation in hepatocellular carcinoma[1][2][3]. |
| Purity | 98.90% |
| MWt | 417.54 |
| Formula | C₂₇H₃₁NO₃ |