GR-73632
GR-73632 is a potent and selective tachykinin NK1 receptor agonist (EC50 = 2 nM in guinea pig vas deferens).
| Supplier | Ace Therapeutics |
|---|---|
| Product # | SMD220 |
| CAS # | 133156-06-6 |
| Pricing | Customizable size, Inquiry |
| Synonym | GR-73632; GR 73632; GR73632. delta-Aminovaleryl-9-pro-10-meleu-substance P (7-10) |
| Product Category | Lab-use Small Molecule Drugs |
| Chemical Formula | C40H59N7O6S |
| Exact Mass | 765.4248 |
| Molecular Weight | 766.015 |
| Elemental Analysis | C, 62.72; H, 7.76; N, 12.80; O, 12.53; S, 4.19 |
| IUPAC/Chemical Name | L-Methioninamide, N-(5-amino-1-oxopentyl)-L-phenylalanyl-L-phenylalanyl-L-prolyl-N-methyl-L-leucyl- |
| InChi Key | HQKPTSSZOJLFBZ-LJADHVKFSA-N |
| InChi Code | InChI=1S/C40H59N7O6S/c1-27(2)24-34(38(51)44-30(36(42)49)20-23-54-4)46(3)40(53)33-18-13-22-47(33)39(52)32(26-29-16-9-6-10-17-29)45-37(50)31(25-28-14-7-5-8-15-28)43-35(48)19-11-12-21-41/h5-10,14-17,27,30-34H,11-13,18-26,41H2,1-4H3,(H2,42,49)(H,43,48)(H,44,51)(H,45,50)/t30-,31-,32-,33-,34-/m0/s1 |
| SMILES Code | CSCC[C@@H](C(N)=O)NC([C@H](CC(C)C)N(C([C@H]1N(C([C@H](CC2=CC=CC=C2)NC([C@H](CC3=CC=CC=C3)NC(CCCCN)=O)=O)=O)CCC1)=O)C)=O |
| Appearance | Solid powder |
| Purity | >95% (or refer to the Certificate of Analysis) |
| Shipping Condition | Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs. |
| Storage Condition | Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years). |
| Solubility | Soluble in DMSO |
| Shelf Life | >2 years if stored properly |
| Drug Formulation | This drug may be formulated in DMSO |
| Stock Solution Storage | 0 - 4℃ for short term (days to weeks), or -20℃ for long term (months). |
| HS Tariff Code | 2934.99.9001 |
| Availability | 2 Weeks |