GKI-1
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-100521-10 mM * 1 mL |
| CAS # | 2444764-03-6 |
| Pricing | 10 mM * 1 mL, USD $495.0 |
| Biological Activity | GKI-1 is a Greatwall (GWL) kinase inhibitor with IC50s of 4.9 and 2.5 µM against hGWLFL and hGWL-KinDom, respectively. GKI-1 robustly inhibits ROCK1 with an IC50 of 11 µM, but only weakly affected PKA[1]. |
| Purity | 99.25% |
| MWt | 269.73 |
| Formula | C₁₅H₁₂ClN₃ |