Cobimetinib (GDC-0973)

Cobimetinib (GDC-0973, RG7420) is a potent and highly selective MEK1 inhibitor with IC50 of 4.2 nM, and showing no significant inhibition when tested against a panel of more than 100 of serine-threonine and tyrosine kinases. Cobimetinib induces apoptosis. Phase 3.

• Supplier: Selleck Chemicals
• Product #: S8041
• Sku #: S8041-5mg