Glutaminase-IN-1
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-114334-10 mM * 1 mL |
| CAS # | 2247127-79-1 |
| Pricing | 10 mM * 1 mL, USD $163.0 |
| Synonyms | CB839 derivative |
| MWt | 618.47 |
| Formula | C₂₆H₂₄F₃N₇O₃Se |
| Biological Activity | Glutaminase-IN-1 (CB839 derivative), a CB839 derivative, is an allosteric inhibitor of 1,3,4-selenadiazole-containing kidney-type glutaminase (KGA), with an IC50 of 1 nM. Glutaminase-IN-1 (CB839 derivative) shows improved cellular uptake and antitumor activity. |
| Purity | 98.05% |