Ac-RYYRIK-NH2
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-P1318 |
| CAS # | 200959-48-4 |
| Pricing | inquire |
| Biological Activity | Ac-RYYRIK-NH2 is a potent and partial agonist on ORL1 transfected in CHO cells (Kd=1.5 nM) and behaves as a endogenous ligand of ORL1. Ac-RYYRIK-NH2 is a specific antagonist for the activation of G protein and competitively antagonizes the stimulation of [35S]-GTPgS binding to G proteins by nociceptin/orphanin FQ (noc/OFQ) in membranes and sections of rat brain[1]. |
| MWt | 939.11 |
| Formula | C₄₄H₇₀N₁₄O₉ |