Elpetrigine
Elpetrigine, also known as GW 273293 and JZP-4, is a potent calcium and sodium channel blocker, which is currently being evaluated in patients as an anticonvulsant and mood stabilizer. JZP-4 could have anxiolytic effects in addition to the anticonvulsant, antidepressant and antimania effects reported earlier.
| Supplier | Ace Therapeutics |
|---|---|
| Product # | SMD847 |
| CAS # | 212778-82-0 |
| Pricing | Customizable size, Inquiry |
| Synonym | GW273293; GW-273293; GW 273293; JZP-4; JZP 4; JZP4; Elpetrigine. |
| Product Category | Lab-use Small Molecule Drugs |
| Chemical Formula | C10H7Cl3N4 |
| Exact Mass | 287.9736 |
| Molecular Weight | 289.544 |
| Elemental Analysis | C, 41.48; H, 2.44; Cl, 36.73; N, 19.35 |
| IUPAC/Chemical Name | 3-(2,3,5-trichlorophenyl)pyrazine-2,6-diamine |
| InChi Key | NNXUYJFHOVCRSM-UHFFFAOYSA-N |
| InChi Code | InChI=1S/C10H7Cl3N4/c11-4-1-5(8(13)6(12)2-4)9-10(15)17-7(14)3-16-9/h1-3H,(H4,14,15,17) |
| SMILES Code | NC1=NC(N)=CN=C1C2=CC(Cl)=CC(Cl)=C2Cl |
| Appearance | Solid powder |
| Purity | >98% (or refer to the Certificate of Analysis) |
| Shipping Condition | Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs. |
| Storage Condition | Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years). |
| Solubility | Soluble in DMSO, not in water |
| Shelf Life | >2 years if stored properly |
| Drug Formulation | This drug may be formulated in DMSO |
| Stock Solution Storage | 0 - 4℃ for short term (days to weeks), or -20℃ for long term (months). |
| HS Tariff Code | 2934.99.9001 |