Sigma-1 receptor antagonist 3
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-125820-10 mM * 1 mL |
| CAS # | 1639220-17-9 |
| Pricing | 10 mM * 1 mL, USD $330.0 |
| Biological Activity | Sigma-1 receptor antagonist 3 (compound135) is a potent and selective Sigma-1 (σ1) receptor antagonist with a Ki of 1.14 nM. Sigma-1 receptor antagonist 3 inhibits Human Ether-a-go-go-Related Gene (hERG) with an IC50 of 1.54 μM. Sigma-1 receptor antagonist 3 has the potential for the neuropathic pain[1]. |
| Purity | 99.47% |
| MWt | 363.86 |
| Formula | C₁₉H₂₃ClFN₃O |