GABAA receptor agent 2 TFA
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-135482 |
| CAS # | 1781880-44-1 |
| Pricing | inquire |
| Biological Activity | GABAA receptor agent 2 TFA is a potent and high-affinity GABAA receptor antagonist with an IC50 of 24 nM (human α1β2γ2 GABAA-expressing tsA201 cells) and a Ki of 28 nM (rat GABAA receptors). GABAA receptor agent 2 TFA is inactive against four human GABA transporters (hGAT-1, hBGT-1, hGAT-2, and hGAT-3)[1]. |
| MWt | 433.42 |
| Formula | C₂₂H₂₂F₃N₃O₃ |