Carfenazine free base
Carfenazine, also known as WY-2445, or carphenazine (BAN), also known as carphenazine maleate (USAN) (brand name Proketazine; former developmental code name NSC-71755), is an antipsychotic and tranquilizer of the phenothiazine group that was withdrawn from the market. Carphenazine blocks postsynaptic mesolimbic dopaminergic D1 and D2 receptors in the brain; depresses the release of hypothalamic and hypophyseal hormones and is believed to depress the reticular activating system thus affecting basal metabolism, body temperature, wakefulness, vasomotor tone, and emesis.
| Supplier | Ace Therapeutics |
|---|---|
| Product # | SMD1451 |
| CAS # | 2622-30-2 (free base) |
| Pricing | Customizable size, Inquiry |
| Synonym | NSC-71755; NSC71755; NSC 71755, Carphenazine free base; Proketazine; Proketazine; Procethazine; carphenazine; NSC 71755; WY2445; WY-2445; WY 2445; |
| Product Category | Lab-use Small Molecule Drugs |
| Chemical Formula | C24H31N3O2S |
| Exact Mass | 425.2137 |
| Molecular Weight | 425.59 |
| Elemental Analysis | C, 67.73; H, 7.34; N, 9.87; O, 7.52; S, 7.53 |
| IUPAC/Chemical Name | 1-(10-(3-(4-(2-hydroxyethyl)piperazin-1-yl)propyl)-10H-phenothiazin-2-yl)propan-1-one |
| InChi Key | XZSMZRXAEFNJCU-UHFFFAOYSA-N |
| InChi Code | InChI=1S/C24H31N3O2S/c1-2-22(29)19-8-9-24-21(18-19)27(20-6-3-4-7-23(20)30-24)11-5-10-25-12-14-26(15-13-25)16-17-28/h3-4,6-9,18,28H,2,5,10-17H2,1H3 |
| SMILES Code | CCC(C(C=C1N2CCCN3CCN(CCO)CC3)=CC=C1SC4=C2C=CC=C4)=O |
| Appearance | Solid powder |
| Purity | >98% (or refer to the Certificate of Analysis) |
| Shipping Condition | Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs. |
| Storage Condition | Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years). |
| Solubility | Soluble in DMSO |
| Shelf Life | >3 years if stored properly |
| Drug Formulation | This drug may be formulated in DMSO |
| Stock Solution Storage | 0 - 4℃ for short term (days to weeks), or -20℃ for long term (months). |
| HS Tariff Code | 2934.99.9001 |
| Availability | 2 Weeks |