| Supplier |
Creative Peptides |
| Product # |
R1850 |
| CAS # |
127060-75-7 |
| Pricing |
Inquire
|
| Synonyms |
Nα-Nicotinoyl-Tyr-(Nα-Cbz-Arg)-Lys-His-Pro-Ile
|
| MolecularFormula |
C52H69N13O11
|
| MolecularWeight |
1052.2
|
| Source |
Synthetic
|
| Sequence |
- One Letter Code: YKHPI (Modifications: Tyr-1 = N-α-Nicotinoyl, Lys-2 = Lys-(N-α-Z-Arg))
- Three Letter Code: nicotinoyl-Tyr-Lys(1)-His-Pro-Ile-OH.Cbz-Arg-(1)
|
| ShippingCondition |
Evaluation sample solution : ship with blue ice; All other available size: ship with RT , or blue ice upon request
|
| Explanation |
CGP-42112A is a potent angiotensin II receptor type 2 (AT2 receptor) agonist. It has a role as an angiotensin receptor agonist, a vasodilator agent, an antineoplastic agent, an anti-inflammatory agent and a neuroprotective agent.
|
| ChemicalName |
N6-(((benzyloxy)carbonyl)-L-arginyl)-N2-(nicotinoyl-L-tyrosyl)-L-lysyl-L-histidyl-L-prolyl-L-isoleucine
|
| Activity |
Potent AT2 angiotensin II receptor agonist.
|
| InChIKey |
UXGNARZDONUMMK-LRMQDCNJSA-N
|
| CanonicalSMILES |
CCC(C)C(C(=O)O)NC(=O)C1CCCN1C(=O)C(CC2=CN=CN2)NC(=O)C(CCCCNC(=O)C(CCCN=C(N)N)NC(=O)OCC3=CC=CC=C3)NC(=O)C(CC4=CC=C(C=C4)O)NC(=O)C5=CN=CC=C5
|
| Solubility |
Soluble to 1 mg/ml in water
|
| IsomericSMILES |
CC[C@H](C)[C@@H](C(=O)O)NC(=O)[C@@H]1CCCN1C(=O)[C@H](CC2=CN=CN2)NC(=O)[C@H](CCCCNC(=O)[C@H](CCCN=C(N)N)NC(=O)OCC3=CC=CC=C3)NC(=O)[C@H](CC4=CC=C(C=C4)O)NC(=O)C5=CN=CC=C5
|
| Appearance |
White solid
|
| Purity |
≥95%
|