GW-803430
GW-803430 is a potent, orally active and selective melanin-concentrating hormone receptor 1 (MCH1) antagonist (IC50 = 9.3 nM). GW-803430 displays antiobesity and antidepressant-like effects in rats and mice.
| Supplier | Ace Therapeutics |
|---|---|
| Product # | SMD885 |
| CAS # | 515141-51-2 |
| Pricing | Customizable size, Inquiry |
| Synonym | GW-803430; GW 803430; GW803430. |
| Product Category | Lab-use Small Molecule Drugs |
| Chemical Formula | C25H24ClN3O3S |
| Exact Mass | 481.1227 |
| Molecular Weight | 481.995 |
| Elemental Analysis | C, 62.30; H, 5.02; Cl, 7.35; N, 8.72; O, 9.96; S, 6.65 |
| IUPAC/Chemical Name | 6-(4-Chlorophenyl)-3-[3-methoxy-4-[2-(1-pyrrolidinyl)ethoxy]phenyl]-thieno[3,2-d]pyrimidin-4(3H)-one |
| InChi Key | MWULMTACIBZPGN-UHFFFAOYSA-N |
| InChi Code | InChI=1S/C25H24ClN3O3S/c1-31-22-14-19(8-9-21(22)32-13-12-28-10-2-3-11-28)29-16-27-20-15-23(33-24(20)25(29)30)17-4-6-18(26)7-5-17/h4-9,14-16H,2-3,10-13H2,1H3 |
| SMILES Code | O=C1C2=C(C=C(C3=CC=C(Cl)C=C3)S2)N=CN1C4=CC=C(OCCN5CCCC5)C(OC)=C4 |
| Appearance | Solid powder |
| Purity | >98% (or refer to the Certificate of Analysis) |
| Shipping Condition | Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs. |
| Storage Condition | Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years). |
| Solubility | Soluble in DMSO |
| Shelf Life | >2 years if stored properly |
| Drug Formulation | This drug may be formulated in DMSO |
| Stock Solution Storage | 0 - 4℃ for short term (days to weeks), or -20℃ for long term (months). |
| HS Tariff Code | 2934.99.9001 |
| Availability | 2 Weeks |