Aprocitentan D4
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-15895S |
| Pricing | inquire |
| Biological Activity | Aprocitentan D4 (ACT-132577 D4) is a deuterium labeled Aprocitentan. Aprocitentan is a major and pharmacologically active metabolite of Macitentan. Aprocitentan is dual ETA/ETB antagonist with IC50s of 3.4 nM and 987 nM, and pA2 valus of 6.7 and 5.5, respectively[1]. |
| Synonyms | ACT-132577 D4 |
| MWt | 550.22 |
| Formula | C₁₆H₁₀D₄Br₂N₆O₄S |