VU0134992 hydrochloride
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-122560A-50 mg |
| CAS # | 1052515-91-9 |
| Pricing | 50 mg, USD $380.0 |
| Biological Activity | VU0134992 hydrochloride is the first subtype-preferring, orally active and selective Kir4.1 potassium channel pore blocker, with an IC50 of 0.97 µM. VU0134992 hydrochloride is 9-fold selective for homomeric Kir4.1 over Kir4.1/5.1 concatemeric channels (IC50=9 µM) at -120 mV[1]. |
| Purity | 99.57% |
| MWt | 447.84 |
| Formula | C₂₀H₃₂BrClN₂O₂ |