EPI-001
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-100348-10 mM * 1 mL |
| CAS # | 227947-06-0 |
| Pricing | 10 mM * 1 mL, USD $88.0 |
| Biological Activity | EPI-001, a selective inhibitor of Androgen Receptor (AR), targets transactivation unit 5 (Tau-5) of the AR. EPI-001 can inhibit transactivation of the AR amino-terminal domain (NTD), with an IC50 of ~6 μM. EPI-001 is also a selective modulator of PPARγ. EPI-001 is active against castration-resistant prostate cancer[1][2][3]. |
| Purity | 98.52% |
| MWt | 394.89 |
| Formula | C₂₁H₂₇ClO₅ |